SCHEMBL10260682

SCHEMBL10260682

Cc1ccc(C(C#N)CC(=O)O)cc1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 14/20 0.62
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
GAA P10253 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HTT P42858 1/20 0.43
ACHE P22303 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27973292 0.84 ALDH1A1 (0.54) FFAR1KMT2AKDM4EMAPTGAA
SCHEMBL25525512 0.84 ALDH1A1 (0.54) FFAR1KMT2AKDM4EMAPTGAA
SCHEMBL434696 0.84 ESR1 (0.58) FFAR1KMT2AALDH1A1
SCHEMBL8697129 0.83 KMT2A (0.53) FFAR1KMT2AKDM4EMAPTGAA
SCHEMBL25525517 0.83 KMT2A (0.53) FFAR1KMT2AKDM4EMAPTGAA
SCHEMBL9556420 0.83 FFAR1 (0.51) FFAR1KMT2A
SCHEMBL27862777 0.83 FFAR1 (0.51) FFAR1KMT2A
SCHEMBL1343883 0.83 FFAR1 (0.51) FFAR1KMT2A
SCHEMBL18382535 0.82 FFAR1 (0.60) FFAR1KMT2ALMNAPOLB
SCHEMBL17144644 0.82 FFAR1 (0.44) FFAR1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11136296-B2 Substituted N-arylethyl-2-arylquinoline-4-carboxamides and use thereof BAYER AKTIENGESELLSCHAFT (DE) 2021-10-05 US disclosed
US-20200031775-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2020-01-30 US disclosed
WO-2012011125-A1 AGONISTS OF GPR40 CONNEXIOS LIFE SCIENCES PVT. LTD. (IN) 2012-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200031775-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF AADAC, NAT1, EPX FFAR1 781/4885KMT2A 921/4885KDM4E 594/4885
US-11136296-B2 Substituted N-arylethyl-2-arylquinoline-4-carboxamides and use thereof AADAC, NAT1, EPX FFAR1 781/4885KMT2A 921/4885KDM4E 594/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.