SCHEMBL10265541

SCHEMBL10265541

BCCCCC1(C(=O)O)CCCN1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ARG2 P78540 15/20 0.67
ARG1 P05089 14/20 0.67
CYP2D6 P10635 4/20 0.33
SLC6A2 P23975 4/20 0.33
SLC6A4 P31645 4/20 0.33
SLC6A3 Q01959 4/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15664945 0.81 ARG2 (0.64) ARG2ARG1CYP2D6SLC6A2SLC6A4
SCHEMBL21285674 0.80 ARG2 (1.00) ARG2ARG1
SCHEMBL893861 0.80 ARG2 (1.00) ARG2ARG1
Hydrochloric Acid SCHEMBL894870 0.79 ARG2 (0.97) ARG2ARG1
SCHEMBL30169846 0.78 ARG1 (0.60) ARG2ARG1
SCHEMBL7094527 0.78 ARG2 (0.60) ARG2ARG1CYP2D6SLC6A2SLC6A4
SCHEMBL31042202 0.77 ARG1 (0.59) ARG2ARG1
SCHEMBL31042217 0.77 ARG1 (0.59) ARG2ARG1
SCHEMBL31042229 0.77 ARG1 (0.59) ARG2ARG1
SCHEMBL31042199 0.77 ARG1 (0.59) ARG2ARG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170183362-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS, INCORPORATED 2017-06-29 US disclosed
US-9040703-B2 Inhibitors of arginase and their therapeutic applications MARS, INCORPORATED (US) 2015-05-26 US disclosed
US-20140371175-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS, INCORPORATED 2014-12-18 US disclosed
US-20120083469-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS, INCORPORATED 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170183362-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS ARG1, ARG2, PRMT9 ARG2 2/4885ARG1 1/4885CYP2D6 459/4885
US-20120083469-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS ARG1, ARG2, PRMT9 ARG2 2/4885ARG1 1/4885CYP2D6 459/4885
US-20140371175-A1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS ARG1, ARG2, PRMT9 ARG2 2/4885ARG1 1/4885CYP2D6 459/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.