SCHEMBL10270191

SCHEMBL10270191

Nc1ccc(NCCNc2nc(-c3ccc(C(F)(F)F)cc3)cc3nc(CN4CCOCC4)nn23)nc1N

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.39
FEN1 P39748 2/20 0.39
SCN9A Q15858 2/20 0.38
ABL1 P00519 1/20 0.38
BCR P11274 1/20 0.38
SLC2A1 P11166 2/20 0.36
TRPV1 Q8NER1 2/20 0.36
ADORA1 P30542 1/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
SIGMAR1 Q99720 1/20 0.36
BTK Q06187 1/20 0.35
KDM4E B2RXH2 1/20 0.35
GLA P06280 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HIF1A Q16665 3/20 0.34
EPAS1 Q99814 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12680869 0.90 ALOX5AP (0.37) ALOX5APFEN1SCN9AABL1BCR
SCHEMBL10270755 0.89 SCN9A (0.40) ALOX5APFEN1SCN9AABL1BCR
SCHEMBL3612472 0.83 ABL1 (0.39) ALOX5APFEN1SCN9AABL1BCR
SCHEMBL10270320 0.82 CALCA (0.35) ALDH1A1KDM4ENPC1RAB9A
SCHEMBL10270318 0.81 ALDH1A1 (0.36) ADORA1ALDH1A1KDM4E
SCHEMBL16784812 0.80 ACVR1 (0.39) SCN9AALDH1A1GAAKDM4EGLA
SCHEMBL16784798 0.79 TBK1 (0.37) ADORA1ALDH1A1KDM4EGLANPC1
SCHEMBL3608208 0.77 SLC2A1 (0.47) ALOX5APFEN1SCN9ASLC2A1TRPV1
SCHEMBL3606754 0.77 SCN9A (0.46) ALOX5APFEN1SCN9ASLC2A1TRPV1
SCHEMBL10270558 0.74 KLK7 (0.37) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137188-B1 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES Bayer Pharma AG (DE) 2012-06-06 EP disclosed
WO-2008113469-A2 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-09-25 WO disclosed