SCHEMBL10270746

SCHEMBL10270746

Cc1ccccc1-c1cc2nccn2c(NCCNc2ccc(N)cn2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K2 Q12851 2/20 0.51
CYP1A2 P05177 9/20 0.38
CLK4 Q9HAZ1 8/20 0.38
FLT1 P17948 1/20 0.37
CDK8 P49336 1/20 0.37
CDK9 P50750 1/20 0.37
LIMK1 P53667 1/20 0.37
ROCK1 Q13464 1/20 0.37
CYP3A4 P08684 5/20 0.36
ALDH1A1 P00352 4/20 0.36
HSD17B10 Q99714 3/20 0.36
ALOX15 P16050 2/20 0.36
MAPK1 P28482 2/20 0.36
CYP2C19 P33261 5/20 0.35
USP2 O75604 1/20 0.35
APEX1 P27695 1/20 0.35
CASP7 P55210 1/20 0.35
HRH4 Q9H3N8 3/20 0.34
TSHR P16473 3/20 0.34
LYN P07948 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10270540 0.89 MAP4K2 (0.40) MAP4K2ALDH1A1LYNSRCBTK
SCHEMBL10270541 0.88 MAP4K2 (0.38) MAP4K2CYP1A2CLK4LIMK1CYP3A4
SCHEMBL12680510 0.86 MAP4K2 (0.47) MAP4K2CYP1A2CLK4FLT1CDK8
SCHEMBL10270290 0.83 MAP4K2 (0.40) MAP4K2CLK4ROCK1ALDH1A1HSD17B10
SCHEMBL10270292 0.82 SYK (0.39) MAP4K2CYP1A2CLK4ROCK1MAPK1
SCHEMBL14079524 0.82 MAPK9 (0.34) MAP4K2CYP1A2CLK4LIMK1CYP3A4
SCHEMBL10270304 0.81 SYK (0.36) MAP4K2CLK4ROCK1MAPK1HRH4
SCHEMBL10269928 0.80 HRH4 (0.48) MAP4K2CLK4ROCK1MAPK1HRH4
SCHEMBL10270160 0.79 MAP4K2 (0.54) MAP4K2CYP1A2CLK4ROCK1CYP3A4
SCHEMBL10270744 0.79 MAP4K2 (0.45) MAP4K2CLK4ROCK1CYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137188-B1 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES Bayer Pharma AG (DE) 2012-06-06 EP disclosed
WO-2008113469-A2 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-09-25 WO disclosed