SCHEMBL1027082

SCHEMBL1027082

CC(C)(C)OC(=O)Nc1ccc([N+](=O)[O-])cc1C#Cc1cncc(N(C(=O)O)C(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.37
HTT P42858 1/20 0.37
MMP1 P03956 3/20 0.36
MMP2 P08253 3/20 0.36
MMP9 P14780 3/20 0.36
MMP8 P22894 3/20 0.36
MMP13 P45452 3/20 0.36
NPC1 O15118 2/20 0.35
MAPT P10636 2/20 0.35
RAB9A P51151 2/20 0.35
POLB P06746 2/20 0.35
ALOX5 P09917 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GAA P10253 2/20 0.34
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1027080 1.00 PKM (0.37) PKMHTTMMP1MMP2MMP9
SCHEMBL1023858 0.88 PKM (0.40) PKMHTTMMP1MMP2MMP9
SCHEMBL1023856 0.88 PKM (0.40) PKMHTTMMP1MMP2MMP9
SCHEMBL1024644 0.87 KCNQ4 (0.35)
SCHEMBL2515901 0.85 EGLN2 (0.35)
SCHEMBL13622742 0.85 PKM (0.41) PKMHTTMMP1MMP2MMP9
SCHEMBL1022924 0.84 GAA (0.40) PKMHTTMMP1MMP2MMP9
SCHEMBL1022925 0.84 GAA (0.40) PKMHTTMMP1MMP2MMP9
SCHEMBL13622511 0.76 MMP1 (0.45) PKMHTTMMP1MMP2MMP9
SCHEMBL1025541 0.76 MAPT (0.42) PKMHTTMMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274288-A2 MACROCYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS Incyte Corporation (US) 2011-01-19 EP disclosed