SCHEMBL10272433

SCHEMBL10272433

CCC(=O)NC(C)C(=O)OC

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
BIRC2 Q13490 1/20 0.45
CA14 Q9ULX7 1/20 0.45
CYP2C9 P11712 1/20 0.45
RECQL P46063 2/20 0.44
MAPT P10636 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2081022 1.00 TSHR (0.51) TSHRMEN1KMT2ABIRC2CA14
SCHEMBL25967050 1.00 TSHR (0.51) TSHRMEN1KMT2ABIRC2CA14
SCHEMBL5571259 0.84 METAP2 (0.45) KMT2ACYP2C9L3MBTL1ALDH1A1
SCHEMBL28081927 0.84 METAP2 (0.45) KMT2ACYP2C9L3MBTL1ALDH1A1
SCHEMBL24967456 0.83 CYP2C9 (0.42) TSHRMEN1KMT2ABIRC2CYP2C9
SCHEMBL27393557 0.83 METAP2 (0.44) KMT2ACYP2C9L3MBTL1
SCHEMBL15479034 0.83 TSHR (0.49) TSHRMEN1KMT2ABIRC2CA14
SCHEMBL10986343 0.80 TSHR (0.50) TSHRMEN1KMT2ABIRC2CA14
SCHEMBL20335032 0.80 TSHR (0.50) TSHRMEN1KMT2ABIRC2CA14
SCHEMBL3673892 0.80 TSHR (0.50) TSHRMEN1KMT2ABIRC2CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025011610-A1 AMIDE DERIVATIVE, AND COMPOSITION AND USE THEREOF 深圳市塔吉瑞生物医药有限公司 2025-01-16 WO disclosed
CN-113874080-B IL-17A modulators and uses thereof 戴斯阿尔法公司 2024-09-27 CN disclosed
CN-117820253-A 3, 6-disubstituted benzothiazole compound and synthesis and application thereof 西北农林科技大学 2024-04-05 CN disclosed
WO-2024042018-A1 A TOPICAL COMPOSITION COMPRISING CHLORINE E6 AND ZINC L-PYROGLUTAMATE ZXA GROUP LTD. (BG) 2024-02-29 WO disclosed
EP-4215530-A1 ISOXAZOLINE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS FMC Corporation (US) 2023-07-26 EP disclosed
EP-1957498-B1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE INC (CA) 2017-02-15 EP disclosed
US-8329726-B2 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE INC. (CA) 2012-12-11 US disclosed
US-20120083482-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE INC. 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120083482-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING HGF, MET, KDR TSHR 173/4885MEN1 4271/4885KMT2A 2894/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.