SCHEMBL10272767

SCHEMBL10272767

O=Cc1ccc(Cn2c(=O)[nH]c3ccsc3c2=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
POLB P06746 4/20 0.55
MAPT P10636 3/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
LMNA P02545 1/20 0.55
RXFP1 Q9HBX9 1/20 0.55
GAA P10253 1/20 0.53
HDAC1 Q13547 1/20 0.53
BLM P54132 1/20 0.52
L3MBTL1 Q9Y468 2/20 0.47
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
ADRB2 P07550 1/20 0.43
TP53 P04637 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1064920 0.81 MEN1 (0.67) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL10272797 0.80 ERCC1 (0.49) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL8347755 0.74 ALDH1A1 (0.54) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL12963438 0.72 ALDH1A1 (0.57) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL1063818 0.70 HDAC1 (1.00) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL7017696 0.68 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL7017699 0.68 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL23997231 0.67 ALDH1A1 (0.56) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL2801455 0.66 HTT (0.54) ALDH1A1MAPTLMNAL3MBTL1HPGD
SCHEMBL9396723 0.66 HTT (0.54) ALDH1A1MEN1KMT2APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed
US-7868204-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2011-01-11 US disclosed
US-7595343-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2009-09-29 US disclosed