SCHEMBL10272800

SCHEMBL10272800

COC(=O)c1ccc(CNc2nccc(I)n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
VNN1 O95497 1/20 0.47
PKM P14618 1/20 0.46
LOXL2 Q9Y4K0 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
ALDH1A1 P00352 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SYK P43405 1/20 0.43
HDAC1 Q13547 2/20 0.43
DRD2 P14416 1/20 0.43
TBXA2R P21731 1/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
HDAC3 O15379 1/20 0.43
NCOR1 O75376 1/20 0.43
HDAC2 Q92769 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1064735 0.86 CA1 (0.60) CA1CA2VNN1PKMLOXL2
SCHEMBL14424237 0.84 CA1 (0.49) CA1CA2VNN1PKMLOXL2
SCHEMBL210753 0.84 ALDH1A1 (0.53) CA1CA2VNN1PKMLOXL2
SCHEMBL10272801 0.80 CA1 (0.50) CA1CA2VNN1PKMLOXL2
SCHEMBL1065202 0.77 HDAC3 (0.74) HDAC1HDAC3NCOR1HDAC2HDAC8
SCHEMBL211213 0.76 HDAC1 (0.63) CA1CA2SYKHDAC1LMNA
SCHEMBL14424239 0.75 CA1 (0.48) CA1CA2PKMLOXL2ALDH1A1
SCHEMBL15761765 0.75 CXCR4 (0.66) CA1CA2PKMNPC1RAB9A
SCHEMBL210701 0.75 CLK4 (0.50) CA1CA2LOXL2NPC1RAB9A
SCHEMBL1063561 0.74 CA1 (0.56) CA1CA2LOXL2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed