SCHEMBL10272801

SCHEMBL10272801

COC(=O)c1ccc(CNc2ccnc(I)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
CLK4 Q9HAZ1 6/20 0.49
ROCK1 Q13464 1/20 0.46
ALDH1A1 P00352 2/20 0.46
USP2 O75604 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
MAPK1 P28482 1/20 0.46
CLK1 P49759 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.44
DYRK1A Q13627 3/20 0.44
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
VNN1 O95497 1/20 0.43
DRD2 P14416 1/20 0.42
TBXA2R P21731 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14424239 0.85 CA1 (0.48) CA1CA2CLK4ROCK1ALDH1A1
SCHEMBL210701 0.84 CLK4 (0.50) CA1CA2CLK4ROCK1ALDH1A1
SCHEMBL10272800 0.80 CA1 (0.51) CA1CA2ALDH1A1LOXL2VNN1
SCHEMBL1064735 0.79 CA1 (0.60) CA1CA2ALDH1A1LOXL2VNN1
SCHEMBL209824 0.77 CLK4 (0.74) CLK4ALDH1A1USP2CYP1A2CYP3A4
SCHEMBL210753 0.77 ALDH1A1 (0.53) CA1CA2CLK4ROCK1ALDH1A1
SCHEMBL15761765 0.77 CXCR4 (0.66) CA1CA2ALDH1A1TSHRPKM
SCHEMBL210650 0.76 ACHE (0.67) ALDH1A1TSHR
SCHEMBL17618077 0.76 RAB9A (0.58) CA1CA2LOXL2DRD2TBXA2R
SCHEMBL16264679 0.76 ALDH1A1 (0.62) CA1CA2ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed