SCHEMBL10272821

SCHEMBL10272821

CCOC(=O)[C@@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)[C@H](O)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAOA P21397 1/20 0.43
CYP26A1 O43174 1/20 0.40
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
MLYCD O95822 1/20 0.38
ADRB2 P07550 2/20 0.38
ADRB1 P08588 2/20 0.38
ADRB3 P13945 2/20 0.38
EPHX2 P34913 1/20 0.37
PPARG P37231 1/20 0.37
PPID Q08752 1/20 0.37
PTGS1 P23219 2/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15237902 0.88 LMNA (0.39) LMNACYP1A2CYP3A4MAOANPC1
SCHEMBL10272817 0.85 LMNA (0.48) LMNACYP1A2CYP3A4MAOACYP26A1
SCHEMBL254790 0.80 ANPEP (0.40) PTGS1
SCHEMBL255440 0.73 TAS1R3 (0.48) NPC1RAB9AADRB2ADRB1ADRB3
SCHEMBL255181 0.73 TAS1R3 (0.48) NPC1RAB9AADRB2ADRB1ADRB3
SCHEMBL15237901 0.73 LMNA (0.40) LMNACYP1A2CYP3A4MAOANPC1
SCHEMBL13366139 0.72 NPSR1 (0.56) CYP1A2NPC1RAB9ASMN1; SMN2TP53
SCHEMBL1761476 0.71 TAS1R3 (0.59) LMNANPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL2973497 0.71 EPHX2 (0.45) EPHX2PPARG
SCHEMBL19262602 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed