SCHEMBL10272847

SCHEMBL10272847

COC(=O)Cc1cc(N)ccc1-c1cnccc1C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 4/20 0.41
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
LCK P06239 1/20 0.38
BTK Q06187 1/20 0.38
MAP4K1 Q92918 11/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
SIRT3 Q9NTG7 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14336221 0.84 ALDH1A1 (0.46) KDM4EALDH1A1GLAGAA
SCHEMBL10272852 0.81 PDGFRB (0.43) CYP17A1ALDH1A1GLACYP11B1CYP11B2
SCHEMBL527037 0.81 GAA (0.52) CYP17A1LCKBTKMAP4K1KDM4E
SCHEMBL10273708 0.80 CYP17A1 (0.65) CYP17A1
SCHEMBL502012 0.76 ALDH1A1 (0.45) KDM4EALDH1A1GLAGAA
SCHEMBL13990328 0.75 ALDH1A1 (0.39) KDM4EALDH1A1GLAGAA
SCHEMBL1408363 0.73 ALDH1A1 (0.45) KDM4EALDH1A1GLAGAA
SCHEMBL5687575 0.73 TSHR (0.50) CYP17A1LCKBTKMAP4K1SIRT3
SCHEMBL15434658 0.73 CCNC (0.42) CCNCCDK8KDM4EALDH1A1GLA
SCHEMBL30940160 0.73 ALDH1A1 (0.45) KDM4EALDH1A1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012015723-A1 SULFONAMIDE COMPOUNDS USEFUL AS CYP17 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-02 WO disclosed