SCHEMBL10275897

SCHEMBL10275897

Cc1nc(Nc2ccc(C(=O)O)cc2)c2ncn(-c3ccc(C#N)cc3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
POLB P06746 1/20 0.47
CDK5 Q00535 1/20 0.47
CDK5R1 Q15078 1/20 0.47
PDE4B Q07343 2/20 0.42
PDE4D Q08499 2/20 0.42
BRAF P15056 1/20 0.41
KDR P35968 1/20 0.41
BTK Q06187 1/20 0.40
YTHDC1 Q96MU7 1/20 0.40
PTPN11 Q06124 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
NR1H4 Q96RI1 1/20 0.38
ADORA2A P29274 1/20 0.38
CRHR1 P34998 1/20 0.37
GAA P10253 1/20 0.37
RCE1 Q9Y256 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10313899 0.87 CRHR1 (0.39) NPC1ADORA2ACRHR1
SCHEMBL10313649 0.84 NPC1 (0.47) NPC1POLBCDK5CDK5R1PDE4B
SCHEMBL10276071 0.84 EGFR (0.43) NPC1KDRCRHR1
SCHEMBL10275611 0.78 MAPK14 (0.51) NPC1POLBPDE4BPDE4DKDR
SCHEMBL10275553 0.74 CTSL (0.41) NPC1CRHR1
SCHEMBL17802587 0.70 CFTR (0.57) NPC1POLBCDK5CDK5R1ADORA2A
SCHEMBL5440509 0.69 BRAF (0.52) NPC1POLBPDE4BPDE4DBRAF
SCHEMBL10313811 0.66 MAPT (0.51) NPC1KDRADORA2ACRHR1
SCHEMBL3135979 0.66 PDE4A (0.55) NPC1POLBCDK5CDK5R1PDE4B
SCHEMBL23675268 0.66 HPGD (0.47) PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF XU LIFENG (US) 2012-07-12 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178915-A1 PYRIMIDINE DERIVATIVES AND ANALOGS, PREPARATION METHOD AND USE THEREOF TYMP, TYMS, ADORA3 NPC1 1381/4885POLB 972/4885CDK5 148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.