SCHEMBL10285200

SCHEMBL10285200

CC(C)(C)OC(=O)N(Cc1ccc(O)c(O)c1)C1CCN(CCn2c(=O)ccc3ccc(O)cc32)CC1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.35
CCR5 P51681 1/20 0.35
HTR2A P28223 3/20 0.34
UBE2M P61081 3/20 0.33
DCUN1D1 Q96GG9 3/20 0.33
NR1H4 Q96RI1 1/20 0.33
KCNH2 Q12809 2/20 0.33
OPRM1 P35372 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10285566 0.93 UBE2M (0.36) HSD11B1CCR5HTR2AUBE2MDCUN1D1
SCHEMBL10285204 0.91 KCNH2 (0.42) HTR2AKCNH2OPRM1
SCHEMBL14279739 0.83 NR1H4 (0.40) HSD11B1CCR5HTR2AUBE2MDCUN1D1
SCHEMBL10285880 0.82 UBE2M (0.35) HSD11B1CCR5HTR2AUBE2MDCUN1D1
SCHEMBL2796897 0.80 KCNH2 (0.41) UBE2MDCUN1D1KCNH2
SCHEMBL10285621 0.80 OPRM1 (0.39) CCR5HTR2ANR1H4KCNH2OPRM1
SCHEMBL2800308 0.79 UBE2M (0.42) CCR5UBE2MDCUN1D1NR1H4KCNH2
SCHEMBL2800489 0.79 KCNH2 (0.52) UBE2MDCUN1D1KCNH2OPRM1
SCHEMBL10285355 0.79 DCUN1D1 (0.37) HSD11B1CCR5UBE2MDCUN1D1
SCHEMBL14279427 0.79 KCNH2 (0.37) KCNH2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed