SCHEMBL10285209

SCHEMBL10285209

Cc1cc(=O)n(CCN2CCC(N(Cc3ccc(O)c(O)c3)C(=O)OC(C)(C)C)CC2)c2cc(OC(F)F)ccc12

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.37
HTR2A P28223 16/20 0.35
CCR5 P51681 1/20 0.33
CNR2 P34972 1/20 0.33
NR1H4 Q96RI1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10285574 0.91 KCNH2 (0.37) KCNH2HTR2ACCR5NR1H4
SCHEMBL10285880 0.90 UBE2M (0.35) KCNH2HTR2ACCR5NR1H4
SCHEMBL12000122 0.89 KCNH2 (0.45) KCNH2NR1H4
SCHEMBL10285211 0.86 STAT3 (0.34) KCNH2CCR5NR1H4
SCHEMBL10285621 0.85 OPRM1 (0.39) KCNH2HTR2ACCR5CNR2NR1H4
SCHEMBL10285573 0.83 GPR119 (0.38) KCNH2CCR5NR1H4
SCHEMBL12000105 0.82 KCNH2 (0.46) KCNH2HTR2A
SCHEMBL2796266 0.81 KCNH2 (0.53) KCNH2CNR2
SCHEMBL10285204 0.81 KCNH2 (0.42) KCNH2HTR2A
SCHEMBL10285571 0.81 CNR2 (0.41) KCNH2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed
EP-1900732-A1 NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2008-03-19 EP disclosed