SCHEMBL10285227

SCHEMBL10285227

COc1ccc2ccc(=O)n(CCCC3(C=O)CCN(C(=O)OC(C)(C)C)CC3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.42
PRKDC P78527 2/20 0.42
MTOR P42345 1/20 0.41
ALDH1A1 P00352 4/20 0.38
STS P08842 1/20 0.37
EPHX2 P34913 1/20 0.37
CCR5 P51681 2/20 0.37
HTT P42858 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 3/20 0.37
HPGD P15428 3/20 0.37
TSHR P16473 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
SLC2A1 P11166 1/20 0.36
BACE1 P56817 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14279666 0.87 HTR1A (0.44) PIK3CAPRKDCMTORALDH1A1KDM4E
SCHEMBL2797642 0.84 PIK3CA (0.42) PIK3CAPRKDCMTORALDH1A1HTT
SCHEMBL13264345 0.84 KCNH2 (0.39) KMT2AMTNR1AMTNR1BNPSR1
SCHEMBL14279499 0.82 PIK3CA (0.43) PIK3CAPRKDCMTORALDH1A1STS
SCHEMBL10285202 0.80 KMT2A (0.38) PIK3CAPRKDCKMT2AMTNR1AMTNR1B
SCHEMBL1712574 0.78 PIK3CA (0.41) PIK3CAPRKDCMTORALDH1A1STS
SCHEMBL14279672 0.78 KDM4E (0.53) ALDH1A1CCR5HTTMEN1KMT2A
SCHEMBL13264611 0.77 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL13264451 0.77 SIGMAR1 (0.46) ALDH1A1KMT2AKDM4E
SCHEMBL2796205 0.76 KMT2A (0.44) ALDH1A1HTTMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed