SCHEMBL10285232

SCHEMBL10285232

O=CC1=C(OS(=O)(=O)C(F)(F)F)CCN(Cc2ccccc2)C1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.42
SLC6A5 Q9Y345 1/20 0.39
ERN1 O75460 1/20 0.39
HTR2A P28223 1/20 0.38
DRD2 P14416 2/20 0.36
DRD3 P35462 2/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
PNMT P11086 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19874109 0.85 DRD2 (0.40) HTR2ADRD2DRD3SIGMAR1ALDH1A1
SCHEMBL19874111 0.85 DRD2 (0.40) HTR2ADRD2DRD3SIGMAR1ALDH1A1
SCHEMBL19886482 0.84 DRD2 (0.39) ACHEDRD2DRD3ALDH1A1
SCHEMBL19874416 0.82 DRD2 (0.40) ACHEDRD2DRD3ALDH1A1KDM4E
SCHEMBL1105716 0.81 ACHE (0.41) ACHESLC6A5DRD2DRD3DRD4
SCHEMBL31288161 0.79 DRD2 (0.38) ACHESLC6A5DRD2DRD3DRD1
SCHEMBL19893177 0.79 ADORA1 (0.41) ACHESLC6A5DRD2DRD3SIGMAR1
SCHEMBL2794854 0.77 CHRM2 (0.46) ALDH1A1
SCHEMBL1901800 0.76 MEN1 (0.48) ALDH1A1
SCHEMBL8672493 0.75 HTR6 (0.42) HTR2ADRD2DRD3DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed