SCHEMBL10285242

SCHEMBL10285242

O=c1cnc2ccc(F)cc2n1CC1CCCO1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.57
ALDH1A1 P00352 15/20 0.52
CYP1A2 P05177 14/20 0.52
HSD17B10 Q99714 8/20 0.52
CASP1 P29466 5/20 0.52
CASP7 P55210 4/20 0.52
CLK4 Q9HAZ1 2/20 0.52
MAPK1 P28482 2/20 0.52
TSHR P16473 5/20 0.51
CYP2C19 P33261 4/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
CYP3A4 P08684 7/20 0.49
CYP2C9 P11712 6/20 0.49
HIF1A Q16665 5/20 0.49
GLA P06280 4/20 0.49
HPGD P15428 4/20 0.49
GAA P10253 1/20 0.49
USP2 O75604 2/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19212760 0.86 GRIN2B (0.47) GRIN2BALDH1A1CYP1A2HSD17B10TSHR
SCHEMBL10285609 0.86 CYP1A2 (0.52) GRIN2BALDH1A1CYP1A2HSD17B10CASP1
SCHEMBL10285226 0.83 ALDH1A1 (0.66) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL2798622 0.83 ALDH1A1 (0.43) GRIN2BALDH1A1CYP1A2HSD17B10CASP1
SCHEMBL15760087 0.78 GRIN2B (0.48) GRIN2BALDH1A1CYP1A2HSD17B10CASP1
SCHEMBL15850872 0.76 KCNH2 (0.38) GRIN2BALDH1A1CYP1A2HSD17B10CASP1
SCHEMBL14313795 0.74 CYP11B1 (0.48) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL29489040 0.74 CYP11B1 (0.48) ALDH1A1CYP1A2HSD17B10CASP1CASP7
SCHEMBL18751788 0.73 GRIN2B (0.68) GRIN2BALDH1A1CYP1A2HSD17B10CASP1
SCHEMBL18363368 0.73 GRIN2B (1.00) GRIN2BCYP1A2CYP2C19CYP2C9GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed
EP-1900732-A1 NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2008-03-19 EP disclosed