SCHEMBL10285609

SCHEMBL10285609

Bc1ccc2ncc(=O)n(CC3CCCO3)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 12/20 0.52
ALDH1A1 P00352 12/20 0.52
HSD17B10 Q99714 5/20 0.52
CASP1 P29466 2/20 0.52
CASP7 P55210 2/20 0.52
CLK4 Q9HAZ1 2/20 0.52
MAPK1 P28482 1/20 0.52
TSHR P16473 5/20 0.51
CYP2C19 P33261 4/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
CYP2C9 P11712 6/20 0.49
CYP3A4 P08684 5/20 0.49
HIF1A Q16665 4/20 0.49
GLA P06280 3/20 0.49
HPGD P15428 2/20 0.49
GAA P10253 1/20 0.49
USP2 O75604 2/20 0.46
LMNA P02545 1/20 0.46
KDM4E B2RXH2 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10285242 0.86 GRIN2B (0.57) CYP1A2ALDH1A1HSD17B10CASP1CASP7
SCHEMBL10285226 0.83 ALDH1A1 (0.66) CYP1A2ALDH1A1HSD17B10CASP1CASP7
SCHEMBL15760087 0.78 GRIN2B (0.48) CYP1A2ALDH1A1HSD17B10CASP1CASP7
SCHEMBL19212760 0.71 GRIN2B (0.47) CYP1A2ALDH1A1HSD17B10TSHRCYP2C19
SCHEMBL2798525 0.68 KDM4E (0.43) ALDH1A1HSD17B10HPGDKDM4ENPSR1
SCHEMBL2798622 0.68 ALDH1A1 (0.43) CYP1A2ALDH1A1HSD17B10CASP1MAPK1
SCHEMBL11999989 0.68 ALDH1A1 (0.43) CYP1A2ALDH1A1HSD17B10CASP1CASP7
SCHEMBL16407633 0.67 ALDH1A1 (0.58) CYP1A2ALDH1A1HSD17B10CASP1CASP7
SCHEMBL29987259 0.66 KDM4C (0.54) ALDH1A1HSD17B10TSHRGAAGRIN2B
SCHEMBL29558920 0.66 KDM4C (0.54) ALDH1A1HSD17B10TSHRGAAGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed