SCHEMBL1028889

SCHEMBL1028889

CC(C)(C)N(C(=O)O)c1cc([N+](=O)[O-])ccc1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.49
SMN1; SMN2 Q16637 5/20 0.46
ALDH1A1 P00352 4/20 0.46
TP53 P04637 2/20 0.46
GPR35 Q9HC97 2/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
GAA P10253 3/20 0.45
THRB P10828 1/20 0.45
ERN1 O75460 1/20 0.43
POLB P06746 2/20 0.43
HTT P42858 2/20 0.43
MAPT P10636 3/20 0.42
NR1H4 Q96RI1 2/20 0.42
CXCR1 P25024 1/20 0.41
CXCR2 P25025 1/20 0.41
LMNA P02545 2/20 0.40
HCRTR1 O43613 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1028886 1.00 L3MBTL1 (0.49) L3MBTL1SMN1; SMN2ALDH1A1TP53GPR35
SCHEMBL16735812 0.84 ALDH1A1 (0.44) L3MBTL1ALDH1A1TP53TSHRGAA
SCHEMBL17099460 0.84 ALDH1A1 (0.44) L3MBTL1ALDH1A1TP53TSHRGAA
SCHEMBL3509375 0.84 ALDH1A1 (0.46) L3MBTL1ALDH1A1TP53TSHRGAA
SCHEMBL3509381 0.84 ALDH1A1 (0.46) L3MBTL1ALDH1A1TP53TSHRGAA
SCHEMBL2209277 0.82 ALDH1A1 (0.56) L3MBTL1SMN1; SMN2ALDH1A1MAPK1GAA
SCHEMBL2209281 0.82 ALDH1A1 (0.56) L3MBTL1SMN1; SMN2ALDH1A1MAPK1GAA
SCHEMBL1026262 0.81 ALDH1A1 (0.48) L3MBTL1SMN1; SMN2ALDH1A1TP53HPGD
SCHEMBL1026260 0.81 ALDH1A1 (0.48) L3MBTL1SMN1; SMN2ALDH1A1TP53HPGD
SCHEMBL20494421 0.80 L3MBTL1 (0.56) L3MBTL1SMN1; SMN2ALDH1A1TP53GPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274288-A2 MACROCYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS Incyte Corporation (US) 2011-01-19 EP disclosed