SCHEMBL1026262

SCHEMBL1026262

CC(C)(C)N(C(=O)O)c1ccc([N+](=O)[O-])cc1I

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.48
HTT P42858 3/20 0.45
TP53 P04637 2/20 0.45
KMT2A Q03164 4/20 0.44
MEN1 O00255 2/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
MAPT P10636 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TDP1 Q9NUW8 3/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
HPGD P15428 3/20 0.38
TSHR P16473 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1026260 1.00 ALDH1A1 (0.48) ALDH1A1HTTTP53KMT2AMEN1
SCHEMBL1026412 0.82 KMT2A (0.58) ALDH1A1HTTTP53KMT2AMEN1
SCHEMBL1026410 0.82 KMT2A (0.58) ALDH1A1HTTTP53KMT2AMEN1
SCHEMBL1028889 0.81 L3MBTL1 (0.49) ALDH1A1HTTTP53LMNAPOLB
SCHEMBL1028886 0.81 L3MBTL1 (0.49) ALDH1A1HTTTP53LMNAPOLB
SCHEMBL16735812 0.80 ALDH1A1 (0.44) ALDH1A1HTTTP53KMT2AMEN1
SCHEMBL3509375 0.80 ALDH1A1 (0.46) ALDH1A1HTTTP53KMT2AMEN1
SCHEMBL3509381 0.80 ALDH1A1 (0.46) ALDH1A1HTTTP53KMT2AMEN1
SCHEMBL17099460 0.80 ALDH1A1 (0.44) ALDH1A1HTTTP53KMT2AMEN1
SCHEMBL2209281 0.78 ALDH1A1 (0.56) ALDH1A1HTTKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274288-A2 MACROCYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS Incyte Corporation (US) 2011-01-19 EP disclosed