SCHEMBL1029436

SCHEMBL1029436

CS(=O)(=O)O.O=C1NC(=O)c2c(O)ccc3cccc1c23

nearest known ligand 0.53

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB known ✓ P27338 1/20 0.38
MCL1 known ✓ Q07820 1/20 0.37
EGFR known ✓ P00533 1/20 0.36
PARP1 P09874 1/20 0.53
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
PKM P14618 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
PARG Q86W56 1/20 0.41
ALDH1A1 P00352 4/20 0.41
GAA P10253 3/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
CASP3 P42574 1/20 0.40
MAPT P10636 3/20 0.39
MAOA P21397 3/20 0.39
POLB P06746 2/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1756367 0.91 PARP1 (0.63) PARP1MEN1KMT2APKMSMN1; SMN2
SCHEMBL789453 0.90 PARP1 (0.61) PARP1MEN1KMT2APKMSMN1; SMN2
Trifluoromethanesulfonic Acid SCHEMBL1028232 0.88 PARP1 (0.49) PARP1MEN1KMT2APKMSMN1; SMN2
Phosphoric Acid SCHEMBL7430846 0.85 PARP1 (0.56) PARP1MEN1KMT2APKMSMN1; SMN2
SCHEMBL1895109 0.85 PARP1 (0.74) PARP1MEN1KMT2APKMSMN1; SMN2
SCHEMBL1027364 0.82 KDM4E (0.51) MEN1KMT2ASMN1; SMN2ALDH1A1GAA
SCHEMBL4101252 0.77 PARP1 (0.56) PARP1MEN1KMT2AALDH1A1GAA
SCHEMBL2041353 0.76 PARP1 (0.51) PARP1MEN1KMT2APKMSMN1; SMN2
SCHEMBL21450709 0.75 PARP1 (0.63) PARP1MEN1KMT2APKMSMN1; SMN2
SCHEMBL28149432 0.74 PARP1 (0.67) PARP1MEN1KMT2APKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102759859-B Resin combination, the manufacture method of hardening thing, resin pattern manufacture method, hardening thing and optical component 富士胶片株式会社 2017-10-24 CN disclosed
EP-2384457-A2 COATING COMPOSITIONS AZ Electronic Materials USA Corp. (US) 2011-11-09 EP disclosed
EP-2273968-A1 COMPOSITIONS AND METHODS INCORPORATING PHOTOCATALYSTS THE PROCTER & GAMBLE COMPANY (US) 2011-01-19 EP disclosed
WO-2010055406-A2 COATING COMPOSITIONS AZ ELECTRONIC MATERIALS USA CORP. (US) 2010-05-20 WO disclosed
WO-2009140076-A1 COMPOSITIONS AND METHODS INCORPORATING PHOTOCATALYSTS THE PROCTER & GAMBLE COMPANY (US) 2009-11-19 WO disclosed