SCHEMBL10317110

SCHEMBL10317110

O=C(O)CN(c1ccc2c(ccn2-c2ccc(OC3COC(c4ccccc4)OC3)nn2)c1)S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
KEAP1 Q14145 9/20 0.33
NFE2L2 Q16236 9/20 0.33
POLB P06746 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13390352 0.92 DGAT1 (0.32) DGAT1
SCHEMBL4553681 0.90 KEAP1 (0.34) ALDH1A1KEAP1NFE2L2DGAT1
SCHEMBL3303955 0.86 ALDH1A1 (0.33) ALDH1A1KEAP1NFE2L2
SCHEMBL3303950 0.86 ALDH1A1 (0.33) ALDH1A1KEAP1NFE2L2
SCHEMBL3325950 0.86 ALDH1A1 (0.33) ALDH1A1KEAP1NFE2L2
SCHEMBL3300839 0.86 KEAP1 (0.35) ALDH1A1KEAP1NFE2L2
SCHEMBL3299910 0.85 DGAT1 (0.31) DGAT1
SCHEMBL13390762 0.82 DGAT1 (0.33) DGAT1
SCHEMBL4440902 0.82 KEAP1 (0.43) KEAP1NFE2L2
SCHEMBL3297170 0.81 KEAP1 (0.36) KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121600-B1 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INT (DE) 2012-07-18 EP disclosed