SCHEMBL10318848

SCHEMBL10318848

COc1ccc2c(Oc3ccc(NS(=O)(=O)c4ccccc4OC(F)(F)F)cc3F)ccnc2c1OC

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AXL P30530 20/20 0.60
EGFR P00533 2/20 0.60
MET P08581 2/20 0.60
SRC P12931 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10319147 0.93 AXL (0.59) AXLEGFRMETSRC
SCHEMBL10319931 0.92 AXL (0.61) AXLEGFRMETSRC
SCHEMBL10317123 0.91 AXL (0.62) AXLEGFRMETSRC
SCHEMBL10318130 0.89 AXL (0.75) AXLEGFRMETSRC
SCHEMBL10317984 0.89 AXL (0.56) AXLEGFRMETSRC
SCHEMBL1591652 0.86 AXL (0.79) AXLEGFRMETSRC
SCHEMBL10318460 0.86 AXL (0.66) AXLEGFRMETSRC
SCHEMBL10316992 0.85 AXL (0.69) AXLEGFRMETSRC
SCHEMBL10317543 0.85 AXL (0.75) AXLEGFRMETSRC
SCHEMBL10317731 0.85 AXL (0.68) AXLEGFRMETSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP claimed