SCHEMBL10319147

SCHEMBL10319147

COc1cc(NS(=O)(=O)c2ccccc2OC(F)(F)F)ccc1Oc1ccnc2c(OC)c(OC)ccc12

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AXL P30530 15/20 0.59
EGFR P00533 1/20 0.54
MET P08581 1/20 0.54
SRC P12931 1/20 0.54
ALPL P05186 2/20 0.46
SLC40A1 Q9NP59 1/20 0.46
SLC22A12 Q96S37 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10319931 0.94 AXL (0.61) AXLEGFRMETSRCALPL
SCHEMBL10318848 0.93 AXL (0.60) AXLEGFRMETSRC
SCHEMBL10317984 0.90 AXL (0.56) AXLEGFRMETSRCALPL
SCHEMBL10318062 0.89 AXL (0.76) AXLEGFRMETSRC
SCHEMBL1590945 0.86 AXL (0.78) AXLEGFRMETSRC
SCHEMBL10317123 0.85 AXL (0.62) AXLEGFRMETSRC
SCHEMBL10317382 0.85 AXL (0.60) AXLEGFRMETSRC
SCHEMBL10316949 0.83 AXL (0.63) AXLEGFRMETSRCALPL
SCHEMBL10317543 0.83 AXL (0.75) AXLEGFRMETSRCSLC40A1
SCHEMBL10318287 0.82 AXL (0.77) AXLEGFRMETSRCSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP claimed