SCHEMBL1032022

SCHEMBL1032022

O=Cc1ccc(OC(F)F)c(OCc2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
TACR2 P21452 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.48
ALDH1A1 P00352 3/20 0.48
LMNA P02545 2/20 0.47
GSK3B P49841 1/20 0.47
KDM4E B2RXH2 1/20 0.47
DRD1 P21728 1/20 0.47
AKR1C3 P42330 2/20 0.46
SIRT2 Q8IXJ6 1/20 0.46
POLB P06746 1/20 0.46
UBE2N P61088 1/20 0.46
KMT2A Q03164 1/20 0.46
PDCD1 Q15116 1/20 0.45
CD274 Q9NZQ7 1/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7371323 0.94 MAOA (0.51) MAOAMAOBTACR2SMN1; SMN2ALDH1A1
SCHEMBL29446267 0.87 TACR2 (0.62) MAOAMAOBTACR2SMN1; SMN2ALDH1A1
SCHEMBL584489 0.87 TACR2 (0.62) MAOAMAOBTACR2SMN1; SMN2ALDH1A1
SCHEMBL8889714 0.86 AKR1C3 (0.50) SMN1; SMN2ALDH1A1LMNADRD1AKR1C3
SCHEMBL18002005 0.86 TACR2 (0.68) TACR2SMN1; SMN2ALDH1A1LMNAAKR1C3
SCHEMBL2460248 0.86 TACR2 (0.53) MAOAMAOBTACR2SMN1; SMN2ALDH1A1
SCHEMBL24707029 0.84 NPC1 (0.55) TACR2SMN1; SMN2ALDH1A1LMNADRD1
SCHEMBL18001824 0.84 POLB (0.49) MAOAMAOBSMN1; SMN2ALDH1A1POLB
SCHEMBL3568939 0.83 RAB9A (0.68) SMN1; SMN2ALDH1A1LMNAKDM4EPOLB
SCHEMBL3568942 0.83 RAB9A (0.68) SMN1; SMN2ALDH1A1LMNAKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260108497-A1 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMACEUTICALC., LTD. (JP) 2026-04-23 US disclosed
US-20240148699-A1 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2024-05-09 US disclosed
EP-3777979-B1 ANTI-INFLAMMATORY COMPOUND AND PREPARATION AND USE THEREOF E NITIATE BIOPHARMACEUTICALS HANGZHOU CO LTD (CN) 2024-01-17 EP disclosed
CN-110407741-B Anti-inflammatory compound and preparation and application thereof 启元生物(杭州)有限公司 2023-03-21 CN disclosed
US-11440886-B2 Anti-inflammatory compound, and preparation and use thereof E-nitiate Biopharmaceuticals (Hangzhou) Co., Ltd. (CN) 2022-09-13 US disclosed
US-20220265613-A1 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2022-08-25 US disclosed
CN-113912593-A Deuterated pyridone compound and application thereof 启元生物(杭州)有限公司 2022-01-11 CN disclosed
CN-110294732-B Pharmaceutical compound for treating liver diseases and application thereof 江苏新元素医药科技有限公司 2021-10-26 CN disclosed
CN-113121417-A Novel piperidine derivative and pharmaceutical application thereof 苏州盛迪亚生物医药有限公司 2021-07-16 CN disclosed
EP-3777979-A1 ANTI-INFLAMMATORY COMPOUND AND PREPARATION AND USE THEREOF Vivavision Biotech, Inc. (CN) 2021-02-17 EP disclosed
US-7425567-B2 Piperidine derivative compounds and drugs containing the compounds as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-09-16 US disclosed
US-7425567-B2 Piperidine derivative compounds and drugs containing the compounds as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-09-16 US disclosed
EP-1954684-A2 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION Otsuka Pharmaceutical Co., Ltd. (JP) 2008-08-13 EP disclosed
WO-2008035316-A2 PHOSPHODIESTERASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2008-03-27 WO disclosed
EP-1869054-A2 CONDENSED ISOXALINE DERIVATIVES AS INHIBITORS OF PHOSPHODIESTERASE TYPE-IV Ranbaxy Laboratories Limited (IN) 2007-12-26 EP disclosed
WO-2007058338-A9 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMA CO LTD (JP) 2007-11-01 WO disclosed
WO-2007058338-A2 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-05-24 WO disclosed
WO-2006085212-A2 CONDENSED ISOXALINE DERIVATIVES AS INHIBITORS OF PHOSPHODIESTERASE TYPE-IV RANBAXY LABORATORIES LIMITED (IN) 2006-08-17 WO disclosed
US-20050080107-A1 Piperidine derivative compounds and drugs containing the compounds as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2005-04-14 US disclosed
EP-1481969-A1 PIPERIDINE DERIVATIVE COMPOUNDS AND DRUGS CONTAINING THE COMPOUNDS AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2004-12-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240148699-A1 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION PDE3B, PDE4A, PDE3A MAOA 34/4885MAOB 61/4885TACR2 1228/4885
US-20260108497-A1 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION PDE7B, PDE4B, PDE1B MAOA 126/4885MAOB 61/4885TACR2 1026/4885
US-20050080107-A1 Piperidine derivative compounds and drugs containing the compounds as the active ingredient PDCD4, PDE4B, IRAK4 MAOA 1167/4885MAOB 1214/4885TACR2 3881/4885
US-11440886-B2 Anti-inflammatory compound, and preparation and use thereof PDE4B, PDE4A, PDE7A MAOA 958/4885MAOB 1655/4885TACR2 2267/4885
US-20220265613-A1 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION PDE3B, PDE4A, PDE3A MAOA 40/4885MAOB 80/4885TACR2 1270/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.