SCHEMBL10333320

SCHEMBL10333320

CSc1ccccc1-c1nc2cc(Cl)c(Cl)cc2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.59
RAB9A P51151 5/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
RHEB Q15382 4/20 0.50
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 3/20 0.49
GPR55 Q9Y2T6 1/20 0.49
PRKAG1 P54619 1/20 0.46
PRKAA2 P54646 1/20 0.46
PRKAB1 Q9Y478 1/20 0.46
NPSR1 Q6W5P4 3/20 0.45
MAPT P10636 2/20 0.45
TTR P02766 1/20 0.45
HSP90AA1 P07900 1/20 0.45
ESR1 P03372 1/20 0.44
AMY1A P0DUB6 1/20 0.44
NPBWR1 P48145 1/20 0.44
ALOX5 P09917 1/20 0.43
GAA P10253 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10333346 0.86 ALDH1A1 (0.47) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL10333235 0.81 KDM4E (0.64) NPC1RAB9AALDH1A1KDM4EGPR55
SCHEMBL15876215 0.79 NPC1 (0.62) NPC1RAB9AMEN1KMT2ARHEB
SCHEMBL22955432 0.78 NPC1 (0.61) NPC1RAB9AMEN1KMT2ARHEB
SCHEMBL10736050 0.78 KDM4E (0.46) NPC1RAB9AALDH1A1KDM4EGPR55
SCHEMBL7270979 0.75 ALOX5 (0.51) NPC1RAB9AALDH1A1KDM4EGPR55
SCHEMBL10768962 0.75 HDAC6 (0.63) NPBWR1
SCHEMBL10768955 0.75 HDAC6 (0.50) NPC1RAB9AALDH1A1KDM4ENPSR1
SCHEMBL3090064 0.75 NPC1 (1.00) NPC1RAB9AMEN1KMT2ARHEB
SCHEMBL9000174 0.74 RHEB (0.73) NPC1RAB9AMEN1KMT2ARHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4900751-A 2-Pyridinyl-phenyl-sulphinyl-and-phenyl-thio-benzimidazoles having antiflammatory or gastic acid secretion inhibition activity FISONS PLC (GB) 1990-02-13 US disclosed
EP-0283504-A1 COMPOUNDS FISONS plc (GB) 1988-09-28 EP disclosed
WO-1988002367-A1 COMPOUNDS FISONS PLC (GB) 1988-04-07 WO disclosed
EP-0262845-A1 Heterocyclic substituted azole derivatives FISONS plc (GB) 1988-04-06 EP disclosed