SCHEMBL10340324

SCHEMBL10340324

COc1ccc(OC)c(CC(=O)Nc2ccccc2C(=O)NCCN(C)C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.52
MAPT P10636 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
PTK2 Q05397 1/20 0.51
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
PKM P14618 2/20 0.48
AURKA O14965 1/20 0.48
AURKB Q96GD4 1/20 0.48
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 3/20 0.47
HTT P42858 2/20 0.47
HSD17B10 Q99714 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
RAD52 P43351 2/20 0.47
UHRF1 Q96T88 1/20 0.47
SMARCA2 P51531 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
MAPK8 P45983 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10340246 0.88 MAPT (0.48) TP53MAPTKMT2AMEN1AURKA
SCHEMBL10340313 0.82 ALDH1A1 (0.65) MAPTKMT2AMEN1AURKAAURKB
SCHEMBL8639959 0.82 KDM4E (0.60) TP53MAPTKMT2AMEN1PKM
SCHEMBL1499413 0.77 PTGS2 (0.61) MAPTPTK2KMT2AMEN1ALDH1A1
SCHEMBL15643259 0.76 KMT2A (0.59) MAPTKMT2AMEN1AURKAAURKB
SCHEMBL19427716 0.75 KMT2A (0.69) TP53MAPTKMT2AMEN1ALDH1A1
SCHEMBL19427444 0.74 ALDH1A1 (0.73) MAPTKMT2AMEN1ALDH1A1HSD17B10
SCHEMBL10340325 0.74 TDP1 (0.47) PTK2ALDH1A1RAD52SMARCA2TDP1
SCHEMBL3362006 0.74 ALDH1A1 (0.62) TP53KMT2AMEN1ALDH1A1KDM4E
SCHEMBL8635693 0.73 ALDH1A1 (0.67) TP53KMT2AMEN1PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0169537-B1 2-PHENYLALKYL-3-AMINOALKYL-4(3H)-QUINAZOLINONES, PROCESSES FOR PREPARING THEM, PHARMACEUTICAL COMPOSITIONS AND USE MITSUBISHI KASEI CORPORATION (JP) 1990-01-03 EP disclosed
US-4668682-A CALCIUM ANTAGONISTS, VASODILATORS, HYPOTENSIVE AGENTS MITSUBISHI CHEMICAL INDUSTRIES LIMITED (JP) 1987-05-26 US disclosed
EP-0169537-A2 2-Phenylalkyl-3-aminoalkyl-4(3H)-quinazolinones, processes for preparing them, pharmaceutical compositions and use MITSUBISHI KASEI CORPORATION (JP) 1986-01-29 EP disclosed