SCHEMBL10340313

SCHEMBL10340313

COc1ccc(OC)c(CC(=O)Nc2ccccc2C(=O)O)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.65
KDM4E B2RXH2 2/20 0.65
HSD17B10 Q99714 2/20 0.65
MEN1 O00255 3/20 0.61
KMT2A Q03164 3/20 0.61
HCAR2 Q8TDS4 3/20 0.60
GAA P10253 2/20 0.60
AKR1C3 P42330 1/20 0.55
AKR1C2 P52895 1/20 0.55
AURKA O14965 1/20 0.55
AURKB Q96GD4 1/20 0.55
CHEK1 O14757 1/20 0.54
PIM1 P11309 1/20 0.54
MAPK8 P45983 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
MAPT P10636 1/20 0.53
TSHR P16473 1/20 0.53
HIF1A Q16665 1/20 0.53
GLS O94925 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639959 0.90 KDM4E (0.60) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL10340271 0.86 KDM4E (0.77) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL10340254 0.86 KDM4E (0.63) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL15643259 0.84 KMT2A (0.59) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL10340147 0.84 ALDH1A1 (0.60) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL6183697 0.83 HIF1A (0.69) ALDH1A1HSD17B10MEN1KMT2ASMN1; SMN2
SCHEMBL19427716 0.83 KMT2A (0.69) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL19427444 0.82 ALDH1A1 (0.73) ALDH1A1HSD17B10MEN1KMT2ASMN1; SMN2
SCHEMBL10340324 0.82 TP53 (0.52) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL28618230 0.80 CHEK1 (0.63) ALDH1A1KDM4EHSD17B10MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0169537-B1 2-PHENYLALKYL-3-AMINOALKYL-4(3H)-QUINAZOLINONES, PROCESSES FOR PREPARING THEM, PHARMACEUTICAL COMPOSITIONS AND USE MITSUBISHI KASEI CORPORATION (JP) 1990-01-03 EP disclosed
US-4668682-A CALCIUM ANTAGONISTS, VASODILATORS, HYPOTENSIVE AGENTS MITSUBISHI CHEMICAL INDUSTRIES LIMITED (JP) 1987-05-26 US disclosed
EP-0169537-A2 2-Phenylalkyl-3-aminoalkyl-4(3H)-quinazolinones, processes for preparing them, pharmaceutical compositions and use MITSUBISHI KASEI CORPORATION (JP) 1986-01-29 EP disclosed