SCHEMBL10340588

SCHEMBL10340588

Cc1cccc(-n2ncc(C=O)c2Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.56
RAB9A P51151 6/20 0.56
PAX8 Q06710 1/20 0.56
NPBWR1 P48145 2/20 0.46
MCHR1 Q99705 2/20 0.46
KMT2A Q03164 2/20 0.45
GRM1 Q13255 1/20 0.44
KDM4E B2RXH2 3/20 0.43
HSD17B10 Q99714 3/20 0.43
HTT P42858 2/20 0.43
BLM P54132 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALDH1A1 P00352 4/20 0.41
MAPT P10636 4/20 0.40
TP53 P04637 4/20 0.40
LMNA P02545 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15332027 0.86 NPC1 (0.48) NPC1RAB9APAX8NPBWR1MCHR1
SCHEMBL15332373 0.82 MAPK14 (0.43) NPC1RAB9APAX8HTTCYP1A2
SCHEMBL15330352 0.82 NPBWR1 (0.45) NPC1RAB9APAX8NPBWR1KMT2A
SCHEMBL3321144 0.81 RAB9A (0.49) NPC1RAB9APAX8NPBWR1KMT2A
SCHEMBL29955120 0.79 NPC1 (0.51) NPC1RAB9ANPBWR1MCHR1KMT2A
SCHEMBL15330816 0.78 MAPT (0.54) NPC1RAB9AKMT2AKDM4EHTT
SCHEMBL15331298 0.77 LMNA (0.43) NPC1RAB9ANPBWR1MCHR1KDM4E
SCHEMBL15331012 0.76 ERN1 (0.39) NPBWR1MCHR1NPSR1ALDH1A1
SCHEMBL2554507 0.75 PTGS1 (0.36) NPC1RAB9ANPBWR1MCHR1KMT2A
SCHEMBL15332330 0.74 NPC1 (0.44) NPC1RAB9ANPBWR1MCHR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0177242-B1 POLLEN FORMATION INHIBITING PYRAZOLES ELI LILLY AND COMPANY (US) 1990-01-03 EP disclosed
US-4775409-A PREVENTING POLLEN FORMATION ELI LILLY AND COMPANY (US) 1988-10-04 US disclosed
US-4666504-A HYBRIDS ELI LILLY AND COMPANY (US) 1987-05-19 US disclosed
EP-0177242-A2 Pollen formation inhibiting pyrazoles ELI LILLY AND COMPANY (US) 1986-04-09 EP disclosed