SCHEMBL1034284

SCHEMBL1034284

C=CCc1c(N)nc(N)nc1O

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
IMPDH2 P12268 1/20 0.33
DHFR P00374 1/20 0.33
CDC7 O00311 1/20 0.32
DBF4 Q9UBU7 1/20 0.32
MAPT P10636 1/20 0.31
CYP2D6 P10635 1/20 0.31
SRD5A1 P18405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3800226 0.90 NPSR1 (0.38) NPSR1IMPDH2DHFRCDC7DBF4
SCHEMBL5807749 0.81 NPSR1 (0.47) NPSR1CDC7DBF4MAPT
SCHEMBL28323788 0.76 NPSR1 (0.39) NPSR1IMPDH2CDC7DBF4CYP2D6
SCHEMBL11208926 0.72 DHFR (0.36) DHFR
SCHEMBL486583 0.69 CASP1 (0.46) NPSR1IMPDH2
SCHEMBL369674 0.69 CASP1 (0.40) NPSR1IMPDH2
SCHEMBL4763149 0.68 KDM4E (0.38) NPSR1MAPTSRD5A1
SCHEMBL3803757 0.68 NPSR1 (0.42) NPSR1IMPDH2CDC7DBF4
SCHEMBL9284251 0.68 NPSR1 (0.55) NPSR1IMPDH2CDC7DBF4MAPT
SCHEMBL1032160 0.68 KDM4E (0.36) NPSR1MAPTCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644389-B1 PYRIMIDINE COMPOUNDS HAVING PHOSPHONATE GROUPS AS ANTIVIRAL NUCLEOTIDE ANALOGS ACAD OF SCIENCE CZECH REPUBLIC (CZ) 2011-01-19 EP disclosed
US-20060241081-A1 Novel compounds and methods for therapy INSTITUTE OF ORGANIC CHEMISTRY 2006-10-26 US disclosed
US-7115592-B2 Phosphonate substituted pyrimidine compounds and methods for therapy INSTITUTE OF ORGANIC CHEMISTRY (CZ) 2006-10-03 US disclosed
EP-1644389-A1 PYRIMIDINE COMPOUNDS HAVING PHOSPHONATE GROUPS AS ANTIVIRAL NUCLEOTIDE ANALOGS INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 2006-04-12 EP disclosed
US-20050075318-A1 Novel compounds and methods for therapy INSTITUTE OF ORGANIC CHENISTRY AND BIOCHEMISTRY ACADEMYOF SCIENCES OF THE CZECH REPUBLIC 2005-04-07 US disclosed
WO-2004111064-A1 PYRIMIDINE COMPOUNDS HAVING PHOSPHONATE GROUPS AS ANTIVIRAL NUCLEOTIDE ANALOGS INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY, ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 2004-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050075318-A1 Novel compounds and methods for therapy ZC3HAV1, IFNAR1, EIF2AK2 NPSR1 2453/4885IMPDH2 512/4885DHFR 72/4885
US-20060241081-A1 Novel compounds and methods for therapy ZC3HAV1, IFNAR1, EIF2AK2 NPSR1 2453/4885IMPDH2 512/4885DHFR 72/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.