SCHEMBL1034426

SCHEMBL1034426

N#Cc1cnccc1NC1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.47
ROCK1 Q13464 1/20 0.47
CDC42BPB Q9Y5S2 1/20 0.47
DYRK1A Q13627 1/20 0.42
CTSL P07711 3/20 0.41
CTSB P07858 3/20 0.41
CTSS P25774 3/20 0.41
CTSK P43235 3/20 0.41
AOC1 P19801 3/20 0.41
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
ALOX15 P16050 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PTGS1 P23219 5/20 0.39
PTGS2 P35354 4/20 0.39
PRKCQ Q04759 2/20 0.39
PRKCD Q05655 2/20 0.39
AOC3 Q16853 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1920243 0.89 AOC1 (0.50) ROCK2ROCK1AOC1PTGS1PTGS2
Hydrochloric Acid SCHEMBL3978097 0.88 AOC1 (0.48) ROCK2ROCK1CDC42BPBDYRK1ACTSL
SCHEMBL29580887 0.82 AOC1 (0.41) ROCK2ROCK1AOC1PTGS1PTGS2
SCHEMBL377808 0.78 CTSL (0.42) CTSLCTSBCTSSCTSKCYP1A2
SCHEMBL14046305 0.77 ROCK2 (0.50) ROCK2ROCK1CDC42BPBDYRK1AAOC1
Hydrochloric Acid SCHEMBL29882259 0.77 CTSL (0.41) CTSLCTSBCTSSCTSKCYP1A2
SCHEMBL12634150 0.77 ROCK2 (0.50) ROCK2ROCK1CDC42BPBDYRK1AAOC1
SCHEMBL19520790 0.76 AOC1 (0.57) CTSKAOC1PTGS1PTGS2AOC3
Hydrochloric Acid SCHEMBL1878276 0.76 ROCK2 (0.49) ROCK2ROCK1CDC42BPBDYRK1AAOC1
SCHEMBL14046304 0.76 ROCK2 (0.49) ROCK2ROCK1CDC42BPBDYRK1AAOC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276730-A2 CARBAMATE AND UREA INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 Vitae Pharmaceuticals, Inc. (US) 2011-01-26 EP disclosed
WO-2009131669-A2 CARBAMATE AND UREA INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-10-29 WO disclosed