SCHEMBL10345506

SCHEMBL10345506

CC1C(c2ccccc2)SCCN1C=O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.38
BRD4 O60885 1/20 0.35
HTR1A P08908 1/20 0.34
LMNA P02545 4/20 0.34
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 2/20 0.34
RECQL P46063 2/20 0.34
TSHR P16473 1/20 0.34
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
ADORA3 P0DMS8 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA7 P36544 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10345857 0.77 BRD4 (0.34) RIPK1BRD4LMNAALDH1A1RECQL
SCHEMBL10345878 0.70
SCHEMBL10345922 0.68
SCHEMBL10345879 0.68 CHRNB2 (0.35) RIPK1ALDH1A1RECQLTSHRPOLB
SCHEMBL10346170 0.68 MMP1 (0.33) RIPK1ALDH1A1POLBSMN1; SMN2
SCHEMBL27284107 0.66 RIPK1 (0.36) RIPK1BRD4
SCHEMBL10346123 0.66 BRD4 (0.43) RIPK1BRD4LMNAALDH1A1KDM4E
SCHEMBL10715111 0.66 USP2 (0.33) BRD4LMNAALDH1A1POLBMAPT
SCHEMBL18065233 0.66
SCHEMBL10346146 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0248854-B1 NOVEL BISPHOSPHONIC DERIVATIVES, A METHOD FOR THEIR PRODUCTION AND A PHARMACEUTICAL COMPOSITION LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 1990-04-25 EP disclosed
US-4870063-A Bisphosphonic acid derivatives, their production and use LEO PHARMACEUTICAL PRODUCTS LTD. A/S (DK) 1989-09-26 US disclosed