SCHEMBL10347983

SCHEMBL10347983

COc1ccc(CO[C@@H]2[C@H](O)C[C@H](OC)O[C@H]2C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
MAPT P10636 1/20 0.39
GJB2 P29033 1/20 0.39
GJA1 P17302 1/20 0.39
TACR1 P25103 1/20 0.37
IDO1 P14902 2/20 0.37
AGXT P21549 2/20 0.37
NAAA Q02083 1/20 0.37
SLC5A2 P31639 3/20 0.37
SLC5A1 P13866 2/20 0.37
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
CYP2D6 P10635 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
HIF1A Q16665 1/20 0.35
MEN1 O00255 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10348013 0.85 REN (0.39) KDM4EMAPTGJB2GJA1TACR1
SCHEMBL16154920 0.80 KDM4E (0.37) KDM4EMAPTGJB2GJA1TACR1
SCHEMBL17898753 0.79 IDO1 (0.42) KDM4EMAPTGJB2GJA1TACR1
SCHEMBL15937685 0.78 IDO1 (0.41) KDM4EMAPTGJB2GJA1TACR1
SCHEMBL8006235 0.75 SLC5A1 (0.42) MAPTGJB2GJA1TACR1IDO1
SCHEMBL8006236 0.75 SLC5A1 (0.42) MAPTGJB2GJA1TACR1IDO1
SCHEMBL8008165 0.75 SLC5A1 (0.42) MAPTGJB2GJA1TACR1IDO1
SCHEMBL8398372 0.75 LGALS8 (0.42) GJB2GJA1TACR1IDO1AGXT
SCHEMBL13380987 0.74 NPC1 (0.45) SLC5A2SLC5A1
SCHEMBL15953973 0.73 IDO1 (0.52) TACR1IDO1AGXTNAAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4962146-A 3-O-glycosyl 16-membered macrolide antibacterials and related derivatives SCHERING CORPORATION (US) 1990-10-09 US disclosed
EP-0362267-A1 3-O-GLYCOSYL 16-MEMBERED MACROLIDE ANTIBACTERIALS AND RELATED DERIVATIVES SCHERING CORPORATION (US) 1990-04-11 EP disclosed
WO-1988008426-A1 3-O-GLYCOSYL 16-MEMBERED MACROLIDE ANTIBACTERIALS AND RELATED DERIVATIVES SCHERING CORPORATION (US) 1988-11-03 WO disclosed