SCHEMBL1034849

SCHEMBL1034849

NS(=O)(=O)c1csc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 8/20 0.51
CA1 P00915 7/20 0.51
CA9 Q16790 5/20 0.49
CA12 O43570 4/20 0.49
CYP2A6 P11509 3/20 0.46
LDHA P00338 1/20 0.46
CA4 P22748 3/20 0.43
CA6 P23280 3/20 0.42
CA5A P35218 2/20 0.42
CA7 P43166 2/20 0.42
CA5B Q9Y2D0 2/20 0.42
CYP2C9 P11712 1/20 0.42
CA14 Q9ULX7 1/20 0.42
MAPT P10636 2/20 0.41
CDK2 P24941 1/20 0.41
PDPK1 O15530 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31287752 1.00 CA2 (0.51) CA2CA1CA9CA12CYP2A6
SCHEMBL29469856 0.80 CA1 (0.47) CA2CA1CA9CA12CYP2A6
SCHEMBL7491058 0.80 CYP2A6 (0.46) CA2CA1CA9CA12CYP2A6
SCHEMBL14089195 0.80 CYP2A6 (0.46) CA2CA1CA9CA12CYP2A6
SCHEMBL2703947 0.80 CYP2A6 (0.47) CA2CA1CA9CA12CYP2A6
SCHEMBL288542 0.80 CA1 (0.47) CA2CA1CA9CA12CYP2A6
Hydrochloric Acid SCHEMBL27734063 0.78 CYP2A6 (0.46) CA2CA1CA9CA12CYP2A6
SCHEMBL10580814 0.78 LDHA (0.48) CA2CA1CA9CA12LDHA
SCHEMBL6628789 0.78 CYP2A6 (0.44) CA2CA1CA9CA12CYP2A6
SCHEMBL6766434 0.78 CYP2A6 (0.46) CA2CA1CA9CA12CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110121499-A (aza) indole-, benzothiophene-and benzofuran-3-sulfonamides 优时比制药有限公司 2019-08-13 CN claimed
CN-103108864-A Arylsulfonamides for treatment of CNS disorders ADAMED SP ZOO 2013-05-15 CN claimed
EP-2493459-A1 OCULAR DRUG DELIVERY DEVICES Aton Pharma, Inc. (US) 2012-09-05 EP claimed
EP-1879877-A2 ANTIMICROBIAL AGENTS Ranbaxy Laboratories Limited (IN) 2008-01-23 EP claimed
WO-2006117762-A2 ANTIMICROBIAL AGENTS RANBAXY LABORATORIES LIMITED (IN) 2006-11-09 WO claimed
CN-118852135-A N-acyl sulfonamide compound, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-10-29 CN disclosed
CN-110121499-A (aza) indole-, benzothiophene-and benzofuran-3-sulfonamides 优时比制药有限公司 2019-08-13 CN disclosed
CN-104529999-A Arylosulfonamides for the treatment of CNS diseases ADAMED SP ZOO 2015-04-22 CN disclosed
CN-103108864-A Arylsulfonamides for treatment of CNS disorders ADAMED SP ZOO 2013-05-15 CN disclosed
US-20110275577-A1 METHODS OF TREATING DERMATOLOGIC, GYNECOLOGIC, AND GENITAL DISORDERS WITH CAFFEIC ACID ANALOGS MOLECULIN, LLC (US) 2011-11-10 US disclosed
EP-2276731-A1 2-SULFONYLAMINO-4-HETEROARYL BUTYRAMIDE ANTAGONISTS OF CCR10 Boehringer Ingelheim International GmbH (DE) 2011-01-26 EP disclosed
WO-2009126675-A1 2-SULFONYLAMINO-4-HETEROARYL BUTYRAMIDE ANTAGONISTS OF CCR10 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-15 WO disclosed
WO-2001049685-A2 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 2001-07-12 WO disclosed
EP-1066272-A1 NOVEL COMPOUNDS USEFUL IN THE COMPLEMENT, COAGULAT AND KALLIKREIN PATHWAYS AND METHOD FOR THEIR PREPARATION BIOCRYST PHARMACEUTICALS INC. (US) 2001-01-10 EP disclosed
WO-1998055471-A1 NOVEL COMPOUNDS USEFUL IN THE COMPLEMENT, COAGULAT AND KALLIKREIN PATHWAYS AND METHOD FOR THEIR PREPARATION BIOCRYST PHARMACEUTICALS, INC. (US) 1998-12-10 WO disclosed
EP-0560554-A2 Antitumor compositions and methods of treatment ELI LILLY AND COMPANY (US) 1993-09-15 EP disclosed
US-5169860-A Benzofuran or benzothiophene arylsulfonylureas ELI LILLY AND COMPANY (US) 1992-12-08 US disclosed
EP-0045196-B1 HERBICIDAL BENZOTHIOPHENE AND BENZOFURAN SULFONAMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-11-13 EP disclosed
US-4391627-A Herbicidal benzothiophene and benzofuran sulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1983-07-05 US disclosed
EP-0045196-A2 Herbicidal benzothiophene and benzofuran sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-02-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110275577-A1 METHODS OF TREATING DERMATOLOGIC, GYNECOLOGIC, AND GENITAL DISORDERS WITH CAFFEIC ACID ANALOGS VHL, PRKDC, POLR1C CA2 581/4885CA1 440/4885CA9 365/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.