SCHEMBL10364211

SCHEMBL10364211

CNC(=O)Nc1cccc(C)c1C(=O)OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
RECQL P46063 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
MAPT P10636 1/20 0.52
DDX3X O00571 2/20 0.47
CISD2 Q8N5K1 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
POLB P06746 3/20 0.45
TDP1 Q9NUW8 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2624007 0.83 ALDH1A1 (0.65) ALDH1A1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL10364587 0.83 NPC1 (0.49) ALDH1A1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL10362887 0.82 NPC1 (0.48) ALDH1A1NPC1RAB9AMAPTDDX3X
SCHEMBL8369698 0.81 ALDH1A1 (0.76) ALDH1A1RECQLSMN1; SMN2NPC1RAB9A
SCHEMBL10362722 0.79 POLB (0.57) ALDH1A1NPC1RAB9AMAPTPOLB
SCHEMBL403705 0.78 CA12 (0.64) ALDH1A1RAB9AMAPTCISD2CA12
SCHEMBL3529435 0.77 KDM4E (0.46) ALDH1A1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL70172 0.75 CA12 (0.59) RAB9AMAPTCA12CA1CA2
SCHEMBL14401688 0.75 ALDH1A1 (0.60) ALDH1A1RECQLSMN1; SMN2NPC1RAB9A
SCHEMBL9686399 0.75 ALDH1A1 (0.60) ALDH1A1RECQLSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0147211-B1 4H-3,1-BENZOXAZIN-4-ONES AND RELATED COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESSES FOR THEIR PREPARATION SYNTEX (U.S.A.) INC. (US) 1990-09-12 EP disclosed
US-4657893-A ANTIINFLAMMATORY AGENTS SYNTEX (U.S.A.) INC. (US) 1987-04-14 US disclosed
EP-0147211-A2 4H-3,1-benzoxazin-4-ones and related compounds, pharmaceutical compositions containing them, and processes for their preparation SYNTEX (U.S.A.) INC. (US) 1985-07-03 EP disclosed