SCHEMBL1036489

SCHEMBL1036489

CC(OC(=O)Oc1ccc([N+](=O)[O-])cc1)O[N+](=O)[O-]

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.52
GAA P10253 1/20 0.51
BCL9 O00512 1/20 0.49
CTNNB1 P35222 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.45
ALDH1A1 P00352 3/20 0.45
KMT2A Q03164 4/20 0.44
PKM P14618 1/20 0.44
MGLL Q99685 2/20 0.44
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
NPC1 O15118 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
LMNA P02545 2/20 0.41
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
THRB P10828 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7989561 0.87 HTR2A (0.53) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL15459741 0.87 HTR2A (0.53) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL2232343 0.86 HTR2A (0.48) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL2233659 0.85 HTR2A (0.52) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL1059539 0.84 HTR2A (0.60) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL2235530 0.84 HTR2A (0.54) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL19457107 0.82 HTR2A (0.52) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL23922815 0.82 HTR2A (0.54) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL21097121 0.82 HTR2A (0.54) HTR2AGAABCL9CTNNB1SMN1; SMN2
SCHEMBL21098059 0.82 HTR2A (0.54) HTR2AGAABCL9CTNNB1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049514-B1 NITRATE ESTERS OF PIPERIDINES NOVARTIS AG (CH) 2011-01-26 EP disclosed
US-20090325947-A1 NITRATE ESTERS OF PIPERIDINES NOVARTIS AG (CH) 2009-12-31 US disclosed
US-20090318432-A1 Nitrate esters of aminoalcohols SPEEDEL EXPERIMENTA AG (CH) 2009-12-24 US disclosed
EP-2061751-A1 NITRATE ESTERS OF AMINOALCOHOLS Novartis Ag (CH) 2009-05-27 EP disclosed
EP-2049514-A1 NITRATE ESTERS OF PIPERIDINES Speedel Experimenta AG (CH) 2009-04-22 EP disclosed
WO-2008031811-A1 NITRATE ESTERS OF AMINOALCOHOLS SPEEDEL EXPERIMENTA AG (CH) 2008-03-20 WO disclosed
WO-2008017685-A1 NITRATE ESTERS OF PIPERIDINES SPEEDEL EXPERIMENTA AG (CH) 2008-02-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090318432-A1 Nitrate esters of aminoalcohols NOS2, NOS1, NOS3 HTR2A 3879/4885GAA 3099/4885BCL9 4314/4885
US-20090325947-A1 NITRATE ESTERS OF PIPERIDINES NOS2, NOS1, NOS3 HTR2A 2234/4885GAA 2901/4885BCL9 2967/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.