SCHEMBL10366159

SCHEMBL10366159

CCCc1cc(C(N)=O)ccc1OCCCNc1cnn(C(C)C)c(=O)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BPTF Q12830 1/20 0.40
KDM4E B2RXH2 2/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CNR2 P34972 3/20 0.37
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
PPARG P37231 2/20 0.34
PPARA Q07869 2/20 0.34
PPARD Q03181 1/20 0.34
TOP2A P11388 2/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
MRGPRX1 Q96LB2 1/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
KAT2B Q92831 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10366155 0.96 KDM4E (0.40) BPTFKDM4ERAB9ASMN1; SMN2CNR2
SCHEMBL10366274 0.92 KDM4E (0.41) BPTFKDM4ERAB9ASMN1; SMN2CNR2
SCHEMBL10366527 0.91 KDM4E (0.39) BPTFKDM4ERAB9ASMN1; SMN2CNR2
SCHEMBL10689346 0.91 PPARA (0.34) BPTFCNR2PDE4APDE4BPDE4C
SCHEMBL10368185 0.90 PTGER4 (0.41) BPTFKDM4ERAB9ASMN1; SMN2CNR2
SCHEMBL10368098 0.88 KDM4E (0.43) BPTFKDM4ERAB9ASMN1; SMN2CNR2
SCHEMBL10685216 0.88 SMN1; SMN2 (0.41) BPTFKDM4ERAB9ASMN1; SMN2CNR2
SCHEMBL10684286 0.86 MTNR1A (0.44) BPTFKDM4ERAB9ASMN1; SMN2CNR2
SCHEMBL10680185 0.85 BPTF (0.40) BPTFKDM4ERAB9ASMN1; SMN2CNR2
SCHEMBL10917891 0.84 KDM4E (0.41) BPTFKDM4ERAB9ASMN1; SMN2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4783462-A 3(2H)pyridazinone, and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1988-11-08 US claimed
EP-0193853-A2 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-09-10 EP claimed
EP-0193853-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1990-09-12 EP disclosed
US-4783462-A 3(2H)pyridazinone, and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1988-11-08 US disclosed
EP-0193853-A2 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-09-10 EP disclosed