SCHEMBL10366552

SCHEMBL10366552

O=[N+]([O-])c1cc(Cc2cccnc2)cnc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
POLB P06746 2/20 0.47
CYP11B1 P15538 3/20 0.46
CYP11B2 P19099 3/20 0.46
CDK5 Q00535 1/20 0.46
CDK5R1 Q15078 1/20 0.46
ALDH1A1 P00352 2/20 0.44
NR1D1 P20393 2/20 0.44
NR1H3 Q13133 2/20 0.44
CYP19A1 P11511 1/20 0.44
PIN1 Q13526 2/20 0.41
MAPT P10636 3/20 0.40
GAA P10253 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
CCR6 P51684 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10365051 0.99 HTT (0.46) HTTSMN1; SMN2POLBCYP11B1CYP11B2
SCHEMBL5038066 0.78 PIN1 (0.37) SMN1; SMN2POLBALDH1A1CYP19A1PIN1
SCHEMBL5033869 0.77 PIN1 (0.62) SMN1; SMN2POLBCYP11B1CYP11B2ALDH1A1
SCHEMBL10920095 0.77 ALDH1A1 (0.48) HTTSMN1; SMN2POLBCYP11B1CYP11B2
SCHEMBL11232440 0.76 CYP11B1 (0.49) CYP11B1CYP11B2ALDH1A1RAB9AL3MBTL1
SCHEMBL5547199 0.76 ALDH1A1 (0.40) POLBCYP11B1CYP11B2ALDH1A1PIN1
SCHEMBL10365876 0.75 ALDH1A1 (0.44) HTTSMN1; SMN2POLBCYP11B1CYP11B2
SCHEMBL487814 0.73 PIN1 (0.39) HTTSMN1; SMN2ALDH1A1PIN1MAPT
SCHEMBL19072274 0.73 SMN1; SMN2 (0.40) HTTSMN1; SMN2ALDH1A1PIN1MAPT
SCHEMBL487553 0.73 PIN1 (0.39) HTTSMN1; SMN2ALDH1A1PIN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0244201-B1 3-HYDROXYPYRIDINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1990-09-26 EP disclosed
US-4863933-A HISTAMINE H1 ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1989-09-05 US disclosed
US-4764519-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1988-08-16 US disclosed