SCHEMBL10370342

SCHEMBL10370342

Nc1nn(CCCN2CCC(O)CC2)c2ccc(O)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.39
MCHR2 Q969V1 1/20 0.38
MCHR1 Q99705 1/20 0.38
ESR2 Q92731 1/20 0.35
KCNA3 P22001 1/20 0.34
SPHK1 Q9NYA1 1/20 0.34
WEE1 P30291 1/20 0.34
HRH3 Q9Y5N1 2/20 0.33
ACHE P22303 2/20 0.33
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
LMNA P02545 1/20 0.33
PGR P06401 1/20 0.33
CHRM2 P08172 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
CHRM1 P11229 1/20 0.33
DRD1 P21728 1/20 0.33
TBXA2R P21731 1/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10368895 0.89 CNR2 (0.36) ESR1MCHR2MCHR1ESR2WEE1
SCHEMBL10369154 0.88 ESR1 (0.46) ESR1ESR2ACHECNR2
SCHEMBL11005140 0.87 TDP1 (0.40) MCHR2MCHR1HRH3ACHEHRH1
SCHEMBL10368046 0.86 ESR1 (0.45) ESR1ESR2PTGS1CNR2
SCHEMBL10367554 0.86 ESR1 (0.45) ESR1ESR2PTGS1CNR2
SCHEMBL10370351 0.85 WEE1 (0.46) ESR1ESR2WEE1KCNH2
SCHEMBL10369107 0.84 CNR2 (0.43) ESR1WEE1LMNAKCNH2CNR2
SCHEMBL10831393 0.84 KCNA3 (0.42) MCHR2MCHR1KCNA3DRD3
SCHEMBL10370283 0.83 ESR1 (0.49) ESR1ESR2HRH3ACHECNR2
SCHEMBL10370294 0.78 ESR1 (0.40) ESR1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0090972-B1 INDAZOLE DERIVATIVES Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1990-05-30 EP disclosed
US-4533731-A ANTIINFLAMMATORY AGENTS ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1985-08-06 US disclosed
EP-0090972-A2 Indazole derivatives Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1983-10-12 EP disclosed