SCHEMBL1037294

SCHEMBL1037294

c1ccc2c(c1)CC2CCN1CCN(c2cccc3c2CCOO3)CC1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9178238 1.00
SCHEMBL9467335 0.94 DRD2 (0.45)
SCHEMBL9176453 0.94 DRD2 (0.45)
SCHEMBL9177231 0.93 DRD4 (0.46)
SCHEMBL9180749 0.93 DRD4 (0.46)
SCHEMBL1038532 0.92 HTR2C (0.44)
SCHEMBL9175625 0.92 HTR2C (0.44)
SCHEMBL9466299 0.90 SIGMAR1 (0.47)
SCHEMBL9175522 0.90 SIGMAR1 (0.47)
SCHEMBL9182178 0.89 HTR2C (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009012-A1 METHODS OF SUPPRESSING APPETITE BY THE ADMINISTRATION OF ANTAGONISTS OF THE SEROTONIN HTR1a or HTR2b RECEPTORS OR INHIBITORS OF TPH2 COLUMBIA UNIVERSITY (US) 2011-01-20 WO disclosed