SCHEMBL103741

SCHEMBL103741

COC(=O)c1ccc(N2C[C@@H](C)N(C(=O)OC(C)(C)C)C[C@@H]2C)c(I)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.41
NPC1 O15118 4/20 0.40
KDM4E B2RXH2 3/20 0.40
RAB9A P51151 2/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
ALDH1A1 P00352 2/20 0.40
ALOX15 P16050 2/20 0.39
HSD17B10 Q99714 2/20 0.39
SETD7 Q8WTS6 2/20 0.39
UCHL1 P09936 1/20 0.38
USP30 Q70CQ3 1/20 0.38
HDAC1 Q13547 3/20 0.37
HDAC6 Q9UBN7 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TSHR P16473 1/20 0.37
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL104152 0.87 KDM4E (0.53) GPR119NPC1KDM4ERAB9AMAPT
SCHEMBL106591 0.85 ALDH1A1 (0.41) NPC1KDM4ERAB9AMAPTHPGD
SCHEMBL16549837 0.84 GPR119 (0.39) GPR119NPC1KDM4ERAB9AMAPT
SCHEMBL103405 0.84 KMT2A (0.46) GPR119KDM4EMAPTHPGDALDH1A1
SCHEMBL16549836 0.84 GPR119 (0.39) GPR119NPC1KDM4ERAB9AMAPT
SCHEMBL2683352 0.77 HDAC1 (0.49) GPR119NPC1KDM4ERAB9AMAPT
SCHEMBL103892 0.75 SMN1; SMN2 (0.47) GPR119NPC1KDM4ERAB9AMAPT
SCHEMBL103471 0.73 ALDH1A1 (0.43) NPC1KDM4ERAB9AMAPTHPGD
SCHEMBL20333136 0.73 HDAC1 (0.52) GPR119KDM4EHDAC1HDAC6TSHR
SCHEMBL103470 0.73 ALDH1A1 (0.43) NPC1KDM4ERAB9AMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426113-A1 CARBINOL COMPOUND HAVING HETEROCYCLIC LINKER Kowa Company, Ltd. (JP) 2012-03-07 EP disclosed