SCHEMBL10374129

SCHEMBL10374129

Cc1cccc(-c2ccccc2C(F)(F)F)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.52
CCR8 P51685 1/20 0.52
HSD11B1 P28845 6/20 0.50
KMO O15229 1/20 0.48
ACP1 P24666 1/20 0.46
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HIF1A Q16665 1/20 0.45
HSD17B10 Q99714 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
PTPN1 P18031 2/20 0.45
CTSA P10619 1/20 0.44
TRPA1 O75762 1/20 0.43
TRPM8 Q7Z2W7 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
CTSK P43235 1/20 0.43
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9369446 0.82 CYP1A2 (0.53) HSD11B1KMOCYP1A2CYP3A4ALOX15
SCHEMBL3366336 0.79 BACE1 (0.51) HSD11B1KMOACP1CYP1A2CYP3A4
SCHEMBL8818449 0.78 CYP1A2 (0.50) ACP1CYP1A2CYP3A4ALOX15TSHR
SCHEMBL20782565 0.77 HSD11B1 (0.51) HSD11B1KMOACP1CYP1A2CYP3A4
SCHEMBL25428915 0.76 KMO (0.60) HSD11B1KMOACP1CYP1A2CYP3A4
SCHEMBL8450245 0.76 CCR1 (0.58) CCR1CCR8
SCHEMBL10374376 0.75 CCR1 (0.62) CCR1CCR8
SCHEMBL13556450 0.75 KMO (0.44) HSD11B1KMOACP1CYP1A2CYP3A4
SCHEMBL1107908 0.75 KMO (0.44) HSD11B1KMOACP1CYP1A2CYP3A4
SCHEMBL10755091 0.75 KMO (0.48) HSD11B1KMOACP1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0244130-B1 PROCESS FOR MAKING 6-ARYL-2-METHYL PYRIDINES ROHM AND HAAS COMPANY (US) 1990-01-17 EP disclosed
US-4804761-A Process for making 6-aryl-2-methylpyridines ROHM AND HAAS COMPANY (US) 1989-02-14 US disclosed
EP-0244130-A2 Process for making 6-aryl-2-methyl pyridines ROHM AND HAAS COMPANY (US) 1987-11-04 EP disclosed
EP-0243101-A2 Insecticidal 6-aryl-pyridine thiosemicarbazones ROHM AND HAAS COMPANY (US) 1987-10-28 EP disclosed
US-4696938-A Insecticidal 6-aryl-pyridine thiosemicarbazones ROHM AND HAAS COMPANY (US) 1987-09-29 US disclosed