SCHEMBL10375232

SCHEMBL10375232

O=C(CCl)c1ccc(-c2ccncc2)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
AGTR1 P30556 1/20 0.47
ADH5 P11766 2/20 0.45
GSK3B P49841 3/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SRD5A2 P31213 1/20 0.41
MARS1 P56192 2/20 0.41
MAPK1 P28482 2/20 0.40
ROCK2 O75116 1/20 0.40
RPS6KA5 O75582 1/20 0.40
MAP4K4 O95819 1/20 0.40
PRKACA P17612 1/20 0.40
RPS6KB1 P23443 1/20 0.40
AKT1 P31749 1/20 0.40
AKT2 P31751 1/20 0.40
GSK3A P49840 1/20 0.40
PRKX P51817 1/20 0.40
NEK4 P51957 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10966713 0.83 AKR1C3 (0.49) ADH5GSK3BMAPK1RPS6KA5MAP4K4
SCHEMBL10965375 0.78 GSK3B (0.55) ALDH1A1GSK3BMAPK1ROCK2RPS6KA5
SCHEMBL10376117 0.75 ALDH1A1 (0.38) ALDH1A1KDM4EAGTR1GSK3BMEN1
SCHEMBL8589404 0.75 GSTO1 (0.50) ALDH1A1KDM4EMEN1KMT2AMAPK1
SCHEMBL5005689 0.74 GSK3B (0.59) ALDH1A1GSK3BSRD5A2MAPK1KMO
SCHEMBL29836035 0.74 GSK3B (0.59) ALDH1A1GSK3BSRD5A2MAPK1KMO
SCHEMBL10585776 0.73 ALDH1A1 (0.60) ALDH1A1KDM4EGSK3BMEN1KMT2A
SCHEMBL10170998 0.72 GSK3B (0.56) ALDH1A1KDM4EGSK3BMAPK1TRPA1
Hydrochloric Acid SCHEMBL4898869 0.72 ALDH1A1 (0.58) ALDH1A1KDM4EGSK3BMEN1KMT2A
SCHEMBL8768769 0.71 GSK3B (0.55) ALDH1A1KDM4EGSK3BMAPK1KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0162333-B1 QUINO-BENZOTHIAZINE ANTIBACTERIAL COMPOUNDS ABBOTT LABORATORIES (US) 1990-06-27 EP disclosed
EP-0162333-A1 Quino-benzothiazine antibacterial compounds ABBOTT LABORATORIES (US) 1985-11-27 EP disclosed
US-4540694-A 1-Pyridine substituted quino-benoxazines and antibacterial use ABBOTT LABORATORIES (US) 1985-09-10 US disclosed
US-4529725-A 1-Pyridine substituted quino-benzothiazine ABBOTT LABORATORIES (US) 1985-07-16 US disclosed