SCHEMBL10375833

SCHEMBL10375833

CCCCOc1ccc2c(c1)CC(=O)N2

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 11/20 0.65
MAOA P21397 8/20 0.55
AHR P35869 1/20 0.49
PDE3B Q13370 3/20 0.48
PDE3A Q14432 3/20 0.48
EIF2AK2 P19525 1/20 0.47
NPC1 O15118 1/20 0.47
KDM1A O60341 1/20 0.46
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19606248 0.88 EIF2AK2 (0.64) MAOBMAOAAHREIF2AK2
SCHEMBL689457 0.88 MAOB (0.62) MAOBMAOAAHRPDE3BPDE3A
SCHEMBL12359302 0.87 MAOB (0.70) MAOBMAOAPDE3BPDE3A
SCHEMBL14333290 0.86 MAOB (0.71) MAOBMAOAAHRPDE3BPDE3A
SCHEMBL7404515 0.85 MAOB (0.65) MAOBMAOAAHRPDE3BPDE3A
SCHEMBL13111961 0.83 MAOB (0.65) MAOBMAOAPDE3BPDE3A
SCHEMBL31718445 0.81 MAOB (0.67) MAOBMAOAPDE3BPDE3A
SCHEMBL23097616 0.80 DRD2 (0.56) MAOBMAOAKCNH2
SCHEMBL20214 0.79 PDE3B (0.66) MAOBMAOAAHRPDE3BPDE3A
SCHEMBL31040124 0.79 PDE3B (0.66) MAOBMAOAAHRPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0155828-B1 PROCESS FOR MAKING 2-OXINDOLE-1-CARBOXAMIDES AND INTERMEDIATES THEREFOR PFIZER INC. (US) 1990-09-19 EP disclosed
EP-0156603-B1 3-SUBSTITUTED 2-OXINDOLE-1-CARBOXAMIDES AS ANALGESIC AND ANTI-INFLAMMATORY AGENTS PFIZER INC. (US) 1989-08-23 EP disclosed
EP-0164860-B1 N,3-DISUBSTITUTED 2-OXINDOLE-1-CARBOXAMIDES AS ANALGESIC AND ANTIINFLAMMATORY AGENTS PFIZER INC. (US) 1989-07-05 EP disclosed
EP-0175551-B1 ANALGESIC AND ANTIINFLAMMATORY 1,3-DIACYL-2-OXINDOLE COMPOUNDS PFIZER INC. (US) 1989-05-10 EP disclosed
EP-0153818-B1 1,3-DISUBSTITUTED 2-OXINDOLES AS ANALGESIC AND ANTI-INFLAMMATORY AGENTS PFIZER INC. (US) 1989-03-15 EP disclosed
US-4808601-A Analgesic and antiinflammatory 1,3-diacyl-2-oxindole compounds PFIZER INC. (US) 1989-02-28 US disclosed
US-4752609-A Analgesic and antiinflammatory 1,3-diacyl-2-oxindole compounds PFIZER INC. (US) 1988-06-21 US disclosed
US-4721712-A 1,3-disubstituted 2-oxindoles as analgesic and anti-inflammatory agents PFIZER INC. (US) 1988-01-26 US disclosed
US-4690943-A ENZYME INHIBITOR OF CYCLOOXYGENASE AND LIPOXYGENASE PFIZER INC. (US) 1987-09-01 US disclosed
US-4665194-A ANALGESICS, ANTIINFLAMMATORY AGENTS PFIZER INC. (US) 1987-05-12 US disclosed
US-4658037-A RHEUMATIC DISEASES PFIZER INC. (US) 1987-04-14 US disclosed
US-4652658-A Process for making 2-oxindole-1-carboxamides and intermediates therefor PFIZER INC. (US) 1987-03-24 US disclosed
EP-0175551-A1 Analgesic and antiinflammatory 1,3-diacyl-2-oxindole compounds PFIZER INC. (US) 1986-03-26 EP disclosed
US-4569942-A N,3-Disubstituted 2-oxindole-1-carboxamides as analgesic and antiinflammatory agents PFIZER INC. (US) 1986-02-11 US disclosed
EP-0164860-A1 N,3-disubstituted 2-oxindole-1-carboxamides as analgesic and antiinflammatory agents PFIZER INC. (US) 1985-12-18 EP disclosed
US-4556672-A 3-Substituted 2-oxindole-1-carboxamides as analgesic and anti-inflammatory agents PFIZER INC. (US) 1985-12-03 US disclosed
EP-0156603-A2 3-Substituted 2-oxindole-1-carboxamides as analgesic and anti-inflammatory agents PFIZER INC. (US) 1985-10-02 EP disclosed
EP-0155828-A2 Process for making 2-oxindole-1-carboxamides and intermediates therefor PFIZER INC. (US) 1985-09-25 EP disclosed
EP-0153818-A2 1,3-Disubstituted 2-oxindoles as analgesic and anti-inflammatory agents PFIZER INC. (US) 1985-09-04 EP disclosed