SCHEMBL10388451

SCHEMBL10388451

O=C(Nc1nccs1)C1CN(c2ccccc2)c2ccccc2C1=O

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
ALDH1A1 P00352 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
RECQL P46063 1/20 0.47
RAB9A P51151 2/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
CYP1A2 P05177 1/20 0.44
NPC1 O15118 1/20 0.44
EGFR P00533 1/20 0.44
TSHR P16473 1/20 0.43
AURKA O14965 1/20 0.43
PIM1 P11309 1/20 0.43
CDK2 P24941 1/20 0.43
GSK3B P49841 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10388212 0.74 NPC1 (0.50) ALDH1A1MEN1KMT2ARECQLRAB9A
SCHEMBL913055 0.71 GRM1 (0.51) ALDH1A1MEN1KMT2ARAB9ALMNA
SCHEMBL11534203 0.71 MEN1 (0.45) TDP1ALDH1A1MEN1KMT2ARAB9A
SCHEMBL11840961 0.70 GAA (0.43) ALDH1A1MEN1KMT2ARAB9ALMNA
SCHEMBL10269831 0.68 GRM1 (0.50) TDP1ALDH1A1MEN1KMT2ARECQL
SCHEMBL11778276 0.67 USP2 (0.55) TDP1ALDH1A1MEN1KMT2ARECQL
SCHEMBL11790890 0.67 ALDH1A1 (0.45) TDP1ALDH1A1MEN1KMT2ARECQL
SCHEMBL11088774 0.65 TDP1 (0.47) TDP1ALDH1A1MEN1KMT2ARECQL
SCHEMBL21294480 0.65 ACSS2 (0.55) ALDH1A1MEN1KMT2ARAB9ALMNA
SCHEMBL11791186 0.65 USP2 (0.52) TDP1ALDH1A1MEN1KMT2ARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4966906-A ANTIINFLAMMATORY AGENTS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-10-30 US disclosed
US-4952588-A ANALGESICS, ANTIINFLAMMATORY AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-08-28 US disclosed
EP-0317991-A2 1-Aryl-3-quinoline- and 1-aryl-3-isoquinoline-carboxamides, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-05-31 EP disclosed
US-4786644-A ANALGESICS, ANTIINFLAMMATORY AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-11-22 US disclosed