SCHEMBL1039439

SCHEMBL1039439

COCCCN1CCOc2ccc(CO[C@H]3CN(C(=O)O)C(C(C)(C)C)[C@@H](CNC(=O)COS(C)(=O)=O)[C@@H]3c3ccc(OC)cc3)cc21

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
RORC P51449 8/20 0.32
MAPT P10636 1/20 0.32
TP53 P04637 1/20 0.31
REN P00797 1/20 0.31
NPY5R Q15761 1/20 0.31
KMT2A Q03164 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1040507 0.92 THRB (0.33) RORCMAPTTP53REN
SCHEMBL1037811 0.91 REN (0.33) PIK3CDPIK3CARORCMAPTTP53
SCHEMBL1040351 0.87 REN (0.35) PIK3CDPIK3CAMAPTREN
SCHEMBL3942761 0.86 RORC (0.34) PIK3CDPIK3CARORCMAPTTP53
SCHEMBL1038354 0.85 REN (0.36) PIK3CDPIK3CARORCMAPTREN
SCHEMBL1039437 0.84 AXL (0.36) PIK3CDPIK3CARORCMAPTTP53
SCHEMBL1039533 0.84 RORC (0.33) RORCRENNPY5R
SCHEMBL1037899 0.83 REN (0.31) REN
SCHEMBL1037898 0.83 REN (0.31) REN
SCHEMBL1038043 0.83 RORC (0.32) RORCREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049514-B1 NITRATE ESTERS OF PIPERIDINES NOVARTIS AG (CH) 2011-01-26 EP disclosed