SCHEMBL10397208

SCHEMBL10397208

CC(C)c1nnc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)c1C=CC=O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GCGR P47871 9/20 0.40
PTGS2 P35354 3/20 0.36
MAPK10 P53779 2/20 0.36
MAPK14 Q16539 2/20 0.36
MAPK9 P45984 1/20 0.36
CSNK1D P48730 1/20 0.36
HMGCR P04035 3/20 0.35
ESR1 P03372 1/20 0.35
CHRM1 P11229 1/20 0.35
TBXA2R P21731 1/20 0.35
PDE4A P27815 1/20 0.35
ADRA1A P35348 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10587512 1.00 GCGR (0.40) GCGRPTGS2MAPK10MAPK14MAPK9
SCHEMBL10397209 0.86 GCGR (0.44) GCGRPTGS2MAPK10MAPK14MAPK9
SCHEMBL8949683 0.83 GCGR (0.53) GCGRHMGCRESR1CHRM1TBXA2R
SCHEMBL8846314 0.81 GCGR (0.44) GCGRPTGS2MAPK10MAPK14MAPK9
SCHEMBL10397582 0.81 GCGR (0.40) GCGRPTGS2MAPK10MAPK14MAPK9
SCHEMBL8949786 0.80 GCGR (0.47) GCGRHMGCRESR1CHRM1TBXA2R
SCHEMBL9744058 0.76 GCGR (0.43) GCGRMAPK10MAPK14HMGCRESR1
SCHEMBL9380517 0.75 RXRA (0.47) GCGRHMGCRESR1CHRM1TBXA2R
SCHEMBL10397220 0.74 HMGCR (0.51) GCGRHMGCRESR1CHRM1TBXA2R
SCHEMBL10397221 0.74 HMGCR (0.51) GCGRHMGCRESR1CHRM1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4946841-A INHIBITORS OF HYDROXYMETHYLGLUTARIC ACID-COENZYME A REDUCTASE HOECHST AKTIENGESELLACHAFT (DE) 1990-08-07 US disclosed
EP-0324347-A2 3,5-Dihydroxycarboxylic acids and their derivatives, process for their preparation, their use as medicines, pharmaceutical compositions and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1989-07-19 EP disclosed