SCHEMBL10397209

SCHEMBL10397209

CC(C)c1nnc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)c1C=O

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCGR P47871 13/20 0.44
PTGS2 P35354 3/20 0.42
MAPK10 P53779 2/20 0.39
MAPK14 Q16539 2/20 0.39
MAPK9 P45984 1/20 0.39
CSNK1D P48730 1/20 0.39
ALDH1A1 P00352 1/20 0.36
PTGS1 P23219 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10587512 0.86 GCGR (0.40) GCGRPTGS2MAPK10MAPK14MAPK9
SCHEMBL10397208 0.86 GCGR (0.40) GCGRPTGS2MAPK10MAPK14MAPK9
SCHEMBL8846314 0.85 GCGR (0.44) GCGRPTGS2MAPK10MAPK14MAPK9
SCHEMBL8949603 0.81 GCGR (0.58) GCGRMAPK10MAPK14
SCHEMBL10397582 0.80 GCGR (0.40) GCGRPTGS2MAPK10MAPK14MAPK9
SCHEMBL8878536 0.78 GCGR (0.46) GCGRPTGS2ALDH1A1
SCHEMBL8877859 0.77 GCGR (0.45) GCGR
SCHEMBL8949673 0.77 GCGR (0.50) GCGRMAPK10MAPK14ALDH1A1
SCHEMBL8879706 0.76 GCGR (0.44) GCGR
SCHEMBL8878486 0.76 GCGR (0.44) GCGRPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4946841-A INHIBITORS OF HYDROXYMETHYLGLUTARIC ACID-COENZYME A REDUCTASE HOECHST AKTIENGESELLACHAFT (DE) 1990-08-07 US disclosed
EP-0324347-A2 3,5-Dihydroxycarboxylic acids and their derivatives, process for their preparation, their use as medicines, pharmaceutical compositions and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1989-07-19 EP disclosed