SCHEMBL10397484

SCHEMBL10397484

CN(Cc1ccc2ccccc2c1)C(=O)Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 1/20 0.50
ACHE P22303 1/20 0.49
TRPV1 Q8NER1 2/20 0.47
MGLL Q99685 1/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2A6 P11509 1/20 0.47
SLC6A2 P23975 4/20 0.47
SLC6A4 P31645 4/20 0.47
SLC6A3 Q01959 3/20 0.47
SIGMAR1 Q99720 1/20 0.46
MC4R P32245 1/20 0.46
MC3R P41968 1/20 0.46
KCNH2 Q12809 2/20 0.45
NPC1 O15118 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
PDK1 Q15118 1/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23972322 0.85 SLC6A2 (0.55) PYCR1ACHETRPV1MGLLCYP1A2
SCHEMBL29565966 0.82 SLC6A2 (0.56) PYCR1ACHETRPV1MGLLCYP1A2
SCHEMBL26027596 0.81 TRPV1 (0.51) PYCR1ACHETRPV1MGLLCYP1A2
SCHEMBL4089366 0.80 PSMB5 (0.57) PYCR1ACHETRPV1MGLLCYP1A2
SCHEMBL3369887 0.78 NPC1 (0.66) MGLLNPC1MEN1KMT2A
SCHEMBL17882156 0.77 RIPK1 (0.68)
SCHEMBL29912607 0.77 RIPK1 (0.68)
SCHEMBL17447228 0.76 PYCR1 (0.61) PYCR1CYP1A2CYP2A6SLC6A2SLC6A4
SCHEMBL6417278 0.76 PDPK1 (0.49) PYCR1ACHETRPV1MGLLCYP1A2
SCHEMBL6417280 0.76 PDPK1 (0.49) PYCR1ACHETRPV1MGLLCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4952595-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1990-08-28 US disclosed
EP-0198382-B1 HETEROCYCLIC AMIDE DERIVATIVES BAYER AG (DE) 1989-09-20 EP disclosed
US-4840961-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1989-06-20 US disclosed
EP-0198382-A2 Heterocyclic amide derivatives BAYER AG (DE) 1986-10-22 EP disclosed