SCHEMBL10399320

SCHEMBL10399320

O=C(c1ccccc1)C(O)[C@H]1O[C@H](Br)[C@@](O)(C(=O)c2ccccc2)[C@@]1(O)C(=O)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.36
LMNA P02545 1/20 0.36
CES1 P23141 1/20 0.36
MAPK1 P28482 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
ATM Q13315 1/20 0.33
HIF1A Q16665 2/20 0.32
EPAS1 Q99814 1/20 0.32
ALKBH5 Q6P6C2 1/20 0.32
MDM2 Q00987 1/20 0.31
GSK3B P49841 2/20 0.31
ALDH1A1 P00352 2/20 0.31
TRPA1 O75762 1/20 0.31
PTPN1 P18031 1/20 0.31
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399319 1.00 CES2 (0.36) CES2LMNACES1MAPK1TDP1
SCHEMBL8822163 0.88 CES2 (0.33) CES2LMNACES1MAPK1TDP1
Hydrochloric Acid SCHEMBL28792392 0.86 CES2 (0.36) CES2LMNACES1MAPK1TDP1
SCHEMBL4582857 0.85 CES2 (0.31) CES2LMNACES1
SCHEMBL28945305 0.84 CES1 (0.37) CES2LMNACES1MAPK1TDP1
SCHEMBL11383230 0.83 LMNA (0.36) CES2LMNACES1MAPK1TDP1
SCHEMBL7638594 0.80 HIF1A (0.37) CES2LMNACES1MAPK1TDP1
SCHEMBL10371759 0.80 CES2 (0.33) CES2LMNACES1TDP1L3MBTL1
SCHEMBL8740392 0.80 CTRB1 (0.38) NPC1RAB9AMDM2
SCHEMBL27797096 0.78 CES2 (0.34) CES2LMNACES1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4977144-A ADENOSINE AGONISTS CIBA-GEIGY CORPORATION (US) 1990-12-11 US disclosed
US-4600771-A Process for the preparation of acylated sugars with a glycosidically bonded isothiocyanate group BAYER AKTIENGESELLSCHAFT (DE) 1986-07-15 US disclosed
EP-0065324-A1 1,3-Diazepine compounds THE UNITED STATES OF AMERICA as represented by the Secretary United States Department of Commerce (US) 1982-11-24 EP disclosed
EP-0034424-A2 Seven-membered ring compounds as inhibitors of cytidine deaminase THE UNITED STATES OF AMERICA as represented by the Secretary United States Department of Commerce (US) 1981-08-26 EP disclosed
WO-1981002164-A1 SEVEN-MEMBERED RING COMPOUNDS AS INHIBITORS OF CYTIDINE DEAMINASE US COMMERCE (US) 1981-08-06 WO disclosed
US-4275057-A CANCER AND ANTITUMOR DRUG RESEARCH THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH, EDUCATION AND WELFARE (US) 1981-06-23 US disclosed